Development of chemical probes: Toward the mode of action of a methylene-linked di(aryl acetate) E1

Bioorganic & Medicinal Chemistry - Tập 18 - Trang 4917-4927 - 2010
Mark E.B. Smith1, Richard M. Gunn1,2, Evelyn Rosivatz3, Lok H. Mak3, Rüdiger Woscholski2,3, Helen C. Hailes1
1Department of Chemistry, University College London, 20 Gordon Street, London WC1H OAJ, UK
2Chemical Biology Centre, Imperial College London, UK
3Division of Cell and Molecular Biology, Imperial College London, UK

Tài liệu tham khảo

Wymann, 2005, Curr. Opin. Cell Biol., 17, 141, 10.1016/j.ceb.2005.02.011 Gunn, 2008, J. Chem. Biol., 1, 49, 10.1007/s12154-008-0008-0 Ho, 2009, FEBS J., 276, 4037, 10.1111/j.1742-4658.2009.07112.x Byrne, 2007, Cell. Signal., 19, 321, 10.1016/j.cellsig.2006.07.004 Katsu, 1984, Chem. Pharm. Bull., 32, 4185, 10.1248/cpb.32.4185 Böhmer, 1987, J. Org. Chem., 52, 3200, 10.1021/jo00391a005 Bruno, 1997, J. Org. Chem., 62, 5174, 10.1021/jo970596h Negishi, 1997, J. Org. Chem., 42, 1821, 10.1021/jo00430a041 Molander, 2006, J. Org. Chem., 71, 9198, 10.1021/jo061699f Hofslokken, 1999, Acta Chem. Scand., 53, 258, 10.3891/acta.chem.scand.53-0258 Mincione, 1978, J. Org. Chem., 43, 1829, 10.1021/jo00403a052 Rosivatz, 2006, ACS Chem. Biol., 1, 780, 10.1021/cb600352f Vlahos, 1994, J. Biol. Chem., 269, 5241, 10.1016/S0021-9258(17)37680-9 Schädel, 2002, Heterocycles, 57, 1049, 10.3987/COM-02-9457 Huang, 2003, J. Am. Chem. Soc., 125, 6653, 10.1021/ja035483w Barder, 2005, J. Am. Chem. Soc., 127, 4685, 10.1021/ja042491j Netherton, 2001, Org. Lett., 3, 4295, 10.1021/ol016971g Huo, 2003, Org. Lett., 5, 423, 10.1021/ol0272693 Bruno, 1997, J. Org. Chem., 62, 5174, 10.1021/jo970596h Tamao, 1972, J. Am. Chem. Soc., 94, 4374, 10.1021/ja00767a075 Sonogashira, 1975, Tetrahedron Lett., 16, 4467, 10.1016/S0040-4039(00)91094-3 Kundu, 1992, Chem. Commun., 41, 10.1039/c39920000041 Pangborn, 1996, Organometallics, 15, 1518, 10.1021/om9503712 Beresford, 2006, Org. Biomol. Chem., 4, 2888, 10.1039/B605026N Antczak, 2006, Synthesis, 18, 3080 Byun, 2008, Bioorg. Med. Chem. Lett., 18, 5591, 10.1016/j.bmcl.2008.08.111 Woscholski, R.; Hailes, H. C.; Numbere, M.; Rosivatz, E. PCT Int. Appl., WO 2006097744, 2006. Payne, 2006, J. Chem. Res., 402, 10.3184/030823406777946752 Buehler, 1943, J. Org. Chem., 8, 316, 10.1021/jo01192a003 Kim, 1991, Ind. Eng. Chem. Res., 30, 1151, 10.1021/ie00054a013 Sergeyev, 2003, Helv. Chim. Acta, 86, 750, 10.1002/hlca.200390074 He, 2006, Tetrahedron, 62, 8755, 10.1016/j.tet.2006.06.104 Casiraghi, 1980, Synthesis, 124, 10.1055/s-1980-28942