Design, synthesis, modeling studies and biological evaluation of thiazolidine derivatives containing pyrazole core as potential anti-diabetic PPAR-γ agonists and anti-inflammatory COX-2 selective inhibitors

Bioorganic Chemistry - Tập 82 - Trang 86-99 - 2019
Khaled R. A. Abdellatif1,2, Wael A.A. Fadaly1, Gehan Kamel3, Yaseen A.M.M. Elshaier4, Mohammed A. El‐Magd5
1Pharmaceutical Organic Chemistry Department, Faculty of Pharmacy, Beni-Suef University, Beni-Suef, Egypt
2Pharmaceutical Sciences Department, Ibn Sina National College for Medical Studies, Jeddah 21418, Saudi Arabia
3Pharmacology Department, Faculty of Veterinary, Cairo University, Cairo, Egypt
4Pharmaceutical Organic Chemistry Department, Faculty of Pharmacy, Al-Azhar University, Assuit, 71524, Egypt
5Anatomy Department, Faculty of Veterinary Medicine, Kafrelshiekh University, Kafrelshiekh, 33516, Egypt

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