Design, synthesis, biological evaluation, and molecular modeling studies of quinoline-ferulic acid hybrids as cholinesterase inhibitors

Bioorganic Chemistry - Tập 93 - Trang 103310 - 2019
Jun Mo1, Hongyu Yang1, Tingkai Chen2, Qihang Li1, Hongzhi Lin1, Feng Feng2,3, Wenyuan Liu4, Wei Qu2, Qinglong Guo5, Heng Chi3, Yao Chen6, Haopeng Sun1,3
1Department of Medicinal Chemistry, School of Pharmacy, China Pharmaceutical University, Nanjing 211198, People’s Republic of China
2Department of Natural Medicinal Chemistry, China Pharmaceutical University, Nanjing 211198, People's Republic of China
3Jiangsu Food and Pharmaceuticals Science College, Institute of Food and Pharmaceuticals Research, 223005, People’s Republic of China
4Department of Pharmaceutical Analysis, Key Laboratory of Drug Quality Control and Pharmacovigilance, Ministry of Education, China Pharmaceutical University, Nanjing 210009, People’s Republic of China
5State Key Laboratory of Natural Medicines, Jiangsu Key Laboratory of Carcinogenesis and Intervention, School of Basic Medicine and Clinical Pharmacy, China Pharmaceutical University, Nanjing, 210009, People's Republic of China
6School of Pharmacy, Nanjing University of Chinese Medicine, Nanjing 210023, People's Republic of China

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