Design, synthesis, and structure–activity relationship of novel orally efficacious pyrazole/sulfonamide based dihydroquinoline γ-secretase inhibitors

Bioorganic & Medicinal Chemistry Letters - Tập 19 - Trang 4920-4923 - 2009
Anh P. Truong1, Danielle L. Aubele1, Gary D. Probst1, Martin L. Neitzel1, Chris M. Semko1, Simeon Bowers1, Darren Dressen1, Roy K. Hom1, Andrei W. Konradi1, Hing L. Sham1,2, Albert W. Garofalo1, Pamela S. Keim2, Jing Wu2, Michael S. Dappen2, Karina Wong3, Erich Goldbach3, Kevin P. Quinn3, John-Michael Sauer3, Elizabeth F. Brigham4, William Wallace5
1Department of Medicinal Chemistry, Elan Pharmaceuticals, 800 Gateway Boulevard, South San Francisco, CA 94080, United States
2Department of Process and Analytical Chemistry, Elan Pharmaceuticals, 1000 Gateway Boulevard, South San Francisco, CA 94080, United States
3Department of Lead Finding, Drug Disposition, and Safety Evaluation, Elan Pharmaceuticals, 800 Gateway Boulevard, South San Francisco, CA 94080, United States
4Department of In Vivo Pharmacology, Elan Pharmaceuticals, 800 Gateway Boulevard, South San Francisco, CA 94080, United States
5Department of Biology, Elan Pharmaceuticals, 1000 Gateway Boulevard, South San Francisco, CA 94080, United States

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