Cytotoxic isoquinoline alkaloids from the aerial parts ofCorydalis incisa

Archives of Pharmacal Research - Tập 30 - Trang 151-154 - 2007
Sang Un Choi1, Nam-ln Baek2, Sung-Hoon Kim3, Jae Heon Yang4, Jae Soon Eun4, Tae Yong Shin4, Jong Pil Lim4, Jae Hyeok Lee5, Hoon Jeon4, Mi-Young Yun4, Kang-Hyun Leem6, Hee Wook Park, Dae Keun Kim4
1Korea Research Institute of Chemical Technology, Taejeon, Korea
2Graduate School of Biotechnology & Plant Metabolism Research Center, Kyung-Hee niversity, Suwon, Korea
3Lab. of Angiogenesis and Chemoprevention, Department of Oriental Pathology, College of Oriental Medicine, KyungHee University, Seoul, Korea
4College of Pharmacy, Woosuk University, Samrye, Korea
5Department of Oriental Pharmaceutical Development, Nambu University, Gwangju, Korea
6College of Oriental Medicine, Semyung University, Jechon, Korea

Tóm tắt

Three known isoquinoline alkaloids were isolated from the chloroform-soluble fraction of the methanolic extract of the aerial parts ofCorydalis incisa (Papaveraceae) through repeated column chromatography. Their chemical structures were elucidated as corynoline (1), corynoloxine (2) and 6-oxocorynoline (3) using spectroscopic analysis. Compounds 1-3 exhibited cytotoxicity against human A549, SK-OV-3, SK-MEL-2 and HCT15 tumor cells.

Tài liệu tham khảo

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