Conformer Analysis of a Biological G-Quadruplex Element in the Human c-MYC Promoter by Native Polyacrylamide Gel Electrophoresis

Journal of Analysis and Testing - Tập 5 - Trang 188-194 - 2021
Xiao-Li Hu1, Hong-Yi Cao1, Liang Fang2, Hua Zuo1
1Key Laboratory of Luminescence Analysis and Molecular Sensing (Southwest University), Ministry of Education, College of Pharmaceutical Sciences, Southwest University, Chongqing, China
2Department of Oncology, The Ninth People’s Hospital of Chongqing, Chongqing, China

Tóm tắt

The G-quadruplexes undergo complex folding and conformation exchanges. G-quadruplex stability is substantially influenced by sequence, buffer and temperature. Mutational analysis together with nuclear magnetic resonance spectroscopy (NMR), X-ray crystallography and circular dichroism spectroscopy has been proved to be a powerful approach for G-quadruplex structural analysis. Herein, we used DNA sequence mutation and native polyacrylamide gel electrophoresis to investigate the topology and conformations of a G-quadruplex model molecule Pu18 found in the human c-MYC promoter. The guanines (G6, G9 or G18) which were not contributable to G-tetrad formation in c-MYC Pu18 sequence were mutated to thymine or adenine. We screened the buffer and temperature of gel electrophoresis for Pu18. Gel electrophoresis showed that two of the four conformers of c-MYC Pu18 in 100 mM K+ buffer were resolved, which was in accordance with the conformations as determined by the 1H NMR spectra in previous studies. This technique is expected as a general methodology for its easy operation and low cost to facilitate uncovering more yet unidentified G-quadruplex folds and functions, with the assistance of other analytical methods like NMR, X-ray crystallography and circular dichroism spectroscopy.

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