Clinical and regulatory perspectives on biosimilar therapies and intended copies of biologics in rheumatology

Springer Science and Business Media LLC - Tập 36 Số 5 - Trang 613-625 - 2016
Eduardo Mysler1, Carlos Pineda2, Takahiko Horiuchi3, Ena Singh4, Ehab Mahgoub4, Javier Coindreau5, Ira Jacobs5
1Reumatólogo en Organización Médica de Investigación, Buenos Aires, Argentina
2Instituto Nacional de Rehabilitacion, Mexico City, Mexico
3Kyushu University Beppu Hospital, Beppu, Japan
4Pfizer Inc., Collegeville, PA, USA
5Pfizer Inc, 235 East 42nd Street, New York, NY 10017-5755, USA

Tóm tắt

Từ khóa


Tài liệu tham khảo

Sahoo N, Choudhury K, Manchikanti P (2009) Manufacturing of biodrugs: need for harmonization in regulatory standards. BioDrugs 23:217–229. doi: 10.2165/11317110-000000000-00000

Lee JF, Litten JB, Grampp G (2012) Comparability and biosimilarity: considerations for the healthcare provider. Curr Med Res Opin 28:1053–1058. doi: 10.1185/03007995.2012.686902

Braun J, van den Berg R, Baraliakos X et al (2011) 2010 update of the ASAS/EULAR recommendations for the management of ankylosing spondylitis. Ann Rheum Dis 70:896–904. doi: 10.1136/ard.2011.151027

Smolen JS, Aletaha D, Bijlsma JW et al (2010) Treating rheumatoid arthritis to target: recommendations of an international task force. Ann Rheum Dis 69:631–637. doi: 10.1136/ard.2009.123919

Smolen JS, Landewe R, Breedveld FC et al (2014) EULAR recommendations for the management of rheumatoid arthritis with synthetic and biological disease-modifying antirheumatic drugs: 2013 update. Ann Rheum Dis 73:492–509. doi: 10.1136/annrheumdis-2013-204573

Gossec L, Smolen JS, Gaujoux-Viala C et al (2012) European League Against Rheumatism recommendations for the management of psoriatic arthritis with pharmacological therapies. Ann Rheum Dis 71:4–12. doi: 10.1136/annrheumdis-2011-200350

Stoll ML, Cron RQ (2014) Treatment of juvenile idiopathic arthritis: a revolution in care. Pediatr Rheumatol Online J 12:13. doi: 10.1186/1546-0096-12-13

Strand V, Sharp V, Koenig AS, Park G, Shi Y, Wang B, Zack DJ, Fiorentino D (2012) Comparison of health-related quality of life in rheumatoid arthritis, psoriatic arthritis and psoriasis and effects of etanercept treatment. Ann Rheum Dis 71:1143–1150. doi: 10.1136/annrheumdis-2011-200387

Al Maini M, Adelowo F, Al Saleh J et al (2015) The global challenges and opportunities in the practice of rheumatology: white paper by the World Forum on Rheumatic and Musculoskeletal Diseases. Clin Rheumatol 34:819–829. doi: 10.1007/s10067-014-2841-6

World Health Organization, Expert Committee on Biological Standardization (2009) Guidelines on evaluation of similar biotherapeutic products (SBPs). World Health Organization. http://www.who.int/biologicals/areas/biological_therapeutics/BIOTHERAPEUTICS_FOR_WEB_22APRIL2010.pdf . Accessed 25 June 2015

European Medicines Agency, Committee for Medicinal Products for Human Use (CHMP) (2014) Guideline on similar biological medicinal products containing biotechnology-derived proteins as active substance: non-clinical and clinical issues. European Medicines Agency. http://www.ema.europa.eu/docs/en_GB/document_library/Scientific_guideline/2015/01/WC500180219.pdf . Accessed 25 July 2015

US Food and Drug Administration, Center for Drug Evaluation and Research (2015) Guidance for industry: scientific considerations in demonstrating biosimilarity to a reference product. US Department of Health and Human Services, US Food and Drug Administration, Center for Drug Evaluation and Research (CDER), Center for Biologics Evaluation and Research (CBER). http://www.fda.gov/downloads/Drugs/GuidanceComplianceRegulatoryInformation/Guidances/UCM291128.pdf . Accessed 25 June 2015

Castaneda-Hernandez G, Gonzalez-Ramirez R, Kay J, Scheinberg MA (2015) Biosimilars in rheumatology: what the clinician should know. RMD Open 1:e000010. doi: 10.1136/rmdopen-2014-000010

Dorner T, Kay J (2015) Biosimilars in rheumatology: current perspectives and lessons learnt. Nat Rev Rheumatol 11:713–724. doi: 10.1038/nrrheum.2015.110

Azevedo VF (2013) Biosimilars require scientifically reliable comparative clinical data. Rev Bras Reumatol 53:129–131. doi: 10.1590/S0482-50042013000100013

Schellekens H (2004) How similar do ‘biosimilars’ need to be? Nat Biotechnol 22:1357–1359. doi: 10.1038/nbt1104-1357

Azevedo VF, Galli N, Kleinfelder A, D’Ippolito J, Urbano PC (2015) Etanercept biosimilars. Rheumatol Int 35:197–209. doi: 10.1007/s00296-014-3080-5

Álvarez AAME, Ruiz de Castilla EM, Flores-Murrieta FJ, Hughes J, Azevedo VF (2014) Recommendations for the regulation of biosimilars and their implementation in Latin America. Generics Biosimilars Initiat J (GaBI J) 3:143–148. doi: 10.5639/gabij.2014.0303.032

Castaneda-Hernandez G, Szekanecz Z, Mysler E, Azevedo VF, Guzman R, Gutierrez M, Rodriguez W, Karateev D (2014) Biopharmaceuticals for rheumatic diseases in Latin America, Europe, Russia, and India: innovators, biosimilars, and intended copies. Joint Bone Spine 81:471–477. doi: 10.1016/j.jbspin.2014.03.019

Azevedo VF (2010) Are we prepared to prescribe biosimilars? Rev Bras Reumatol 50:221–224

Dorner T, Strand V, Castaneda-Hernandez G, Ferraccioli G, Isaacs JD, Kvien TK, Martin-Mola E, Mittendorf T, Smolen JS, Burmester GR (2013) The role of biosimilars in the treatment of rheumatic diseases. Ann Rheum Dis 72:322–328. doi: 10.1136/annrheumdis-2012-202715

Yoo DH, Hrycaj P, Miranda P et al (2013) A randomised, double-blind, parallel-group study to demonstrate equivalence in efficacy and safety of CT-P13 compared with innovator infliximab when coadministered with methotrexate in patients with active rheumatoid arthritis: the PLANETRA study. Ann Rheum Dis 72:1613–1620. doi: 10.1136/annrheumdis-2012-203090

Horiuchi T, Mitoma H, Harashima S, Tsukamoto H, Shimoda T (2010) Transmembrane TNF-alpha: structure, function and interaction with anti-TNF agents. Rheumatology (Oxford) 49:1215–1228. doi: 10.1093/rheumatology/keq031

Park W, Hrycaj P, Jeka S et al (2013) A randomised, double-blind, multicentre, parallel-group, prospective study comparing the pharmacokinetics, safety, and efficacy of CT-P13 and innovator infliximab in patients with ankylosing spondylitis: the PLANETAS study. Ann Rheum Dis 72:1605–1612. doi: 10.1136/annrheumdis-2012-203091

Zelenetz AD, Ahmed I, Braud EL et al (2011) NCCN Biosimilars White Paper: regulatory, scientific, and patient safety perspectives. J Natl Compr Cancer Netw 9(Suppl 4):S1–S22

Schellekens H (2009) Biosimilar therapeutics—What do we need to consider? NDT Plus 2:i27–i36. doi: 10.1093/ndtplus/sfn177

Anfinsen CB (1972) The formation and stabilization of protein structure. Biochem J 128:737–749

Pauling L, Corey RB, Branson HR (1951) The structure of proteins; two hydrogen-bonded helical configurations of the polypeptide chain. Proc Natl Acad Sci USA 37:205–211

Alberts B, Johnson A, Lewis J, Raff M, Roberts K, Walters P (2002) The shape and structure of proteins. In: Molecular biology of the cell, 4th edn. Garland Science, New York and London

Creighton TE (1993) Proteins: structures and molecular properties, 2nd edn. Macmillan, New York

Behme S (2015) The manufacturing of pharmaceutical proteins: from technology to economy, 2nd edn. Wiley-VCH, Weinheim

Avis KE, Wu VL (1996) Biotechnology and biopharmaceutical manufacturing, processing, and preservation. CRC Press, Boca Raton

Mellstedt H, Niederwieser D, Ludwig H (2008) The challenge of biosimilars. Ann Oncol 19:411–419. doi: 10.1093/annonc/mdm345

Schneider CK, Kalinke U (2008) Toward biosimilar monoclonal antibodies. Nat Biotechnol 26:985–990. doi: 10.1038/nbt0908-985

Schellekens H (2005) Follow-on biologics: challenges of the “next generation”. Nephrol Dial Transplant 20(Suppl 4):iv31–iv36. doi: 10.1093/ndt/gfh1085

Kuhlmann M, Covic A (2006) The protein science of biosimilars. Nephrol Dial Transplant 21(Suppl 5):v4–v8. doi: 10.1093/ndt/gfl474

Schellekens H (2002) Bioequivalence and the immunogenicity of biopharmaceuticals. Nat Rev Drug Discov 1:457–462. doi: 10.1038/nrd818

Schellekens H (2005) Factors influencing the immunogenicity of therapeutic proteins. Nephrol Dial Transplant 20(Suppl 6):vi3–vi9. doi: 10.1093/ndt/gfh1092

Walsh G (2003) The drug manufacturing process. In: Biopharmaceuticals: biochemistry and biotechnology, 2nd edn. Wiley, Hoboken, pp 93–187

Chirino AJ, Mire-Sluis A (2004) Characterizing biological products and assessing comparability following manufacturing changes. Nat Biotechnol 22:1383–1391. doi: 10.1038/nbt1030

McCamish M, Woollett G (2011) Worldwide experience with biosimilar development. MAbs 3:209–217

ICH Expert Working Group (2004) Comparability of biotechnological/biological products subject to changes in their manufacturing process. In: International conference on harmonisation (ICH) of technical requirements for registration of pharmaceuticals for human use. http://www.ich.org/fileadmin/Public_Web_Site/ICH_Products/Guidelines/Quality/Q5E/Step4/Q5E_Guideline.pdf . Accessed 25 July 2015

Venema J, Tebbey P, Varga A, Naill M, Wang X, Cui L, Clewell J (2015) Humira® (adalimumab): fifteen years of controlled production and consistency of quality attributes. Ann Rheum Dis 72:461

Berkowitz SA, Engen JR, Mazzeo JR, Jones GB (2012) Analytical tools for characterizing biopharmaceuticals and the implications for biosimilars. Nat Rev Drug Discov 11:527–540. doi: 10.1038/nrd3746

Health Canada (2008) Guidance for sponsors: information and submission requirements for subsequent entry biologics (SEBs). Minister of Public Works and Government Services Canada. http://www.hc-sc.gc.ca/dhp-mps/alt_formats/pdf/brgtherap/applic-demande/guides/seb-pbu/seb-pbu-2010-eng.pdf . Accessed 25 July 2015

Dranitsaris G, Dorward K, Hatzimichael E, Amir E (2013) Clinical trial design in biosimilar drug development. Invest New Drugs 31:479–487. doi: 10.1007/s10637-012-9899-2

Alten R, Cronstein B (2015) Clinical trial development for biosimilars. Semin Arthritis Rheum 44:S2–S8. doi: 10.1016/j.semarthrit.2015.04.002

Mysler E (2015) Biosimilars: clinical interpretation and implications for drug development. Curr Rheumatol Rep 17:8. doi: 10.1007/s11926-014-0483-y

Kay J, Smolen J (2013) Biosimilars to treat inflammatory arthritis: the challenge of proving identity. Ann Rheum Dis 72:1589–1593. doi: 10.1136/annrheumdis-2012-203198

Mysler E, Scheinberg M (2012) Biosimilars in rheumatology: a view from Latin America. Clin Rheumatol 31:1279–1280. doi: 10.1007/s10067-012-2068-3

Generics and Biosimilars Initiative (GaBI) (2013) Regulation of similar biotherapeutic products in Latin America. Pro Pharma Communications International. http://www.gabionline.net/Biosimilars/Research/Regulation-of-similar-biotherapeutic-products-in-Latin-America . Accessed 25 July 2015

Castanheira LG, Barbano DB, Rech N (2011) Current development in regulation of similar biotherapeutic products in Brazil. Biologicals 39:308–311. doi: 10.1016/j.biologicals.2011.06.021

Generics and Biosimilars Initiative (GaBI) (2013) Colombia issues draft decree for registration of biologicals. Pro Pharma Communications International. http://www.gabionline.net/Guidelines/Colombia-issues-draft-decree-for-registration-of-biologicals . Accessed 25 July 2015

Desanvicente-Celis Z, Caro-Moreno J, Enciso-Zuluaga M, Anaya JM (2013) Similar biotherapeutic products in Latin America. Regulation and opportunities for patients with autoimmune diseases. Biosimilars 3:1–17. doi: 10.2147/BS.S38572

Espinosa Morales R, Diaz Borjon A, Barile Fabris LA et al (2013) Biosimilar drugs in Mexico: position of the Mexican College of Rheumatology, 2012. Reumatol Clin 9:113–116. doi: 10.1016/j.reuma.2012.11.001

Lapadula G, Ferraccioli GF (2012) Biosimilars in rheumatology: pharmacological and pharmacoeconomic issues. Clin Exp Rheumatol 30:S102–S106

COFEPRIS (2014) La COFEPRIS revoca registro del produco “Kikuzumab”. Federal Commission for the Protection against Sanitary Risk (COFEPRIS), Mexico Department of Health. www.cofepris.gob.mx . Accessed 3 Aug 2015

Azevedo VFSE, Siemak B, Halbert RJ (2012) Potential regulatory and commercial environment for biosimilars in Latin America. Value Health Reg Issues 2:228–234. doi: 10.1016/j.vhri.2012.09.015

World Health Organization (2015) Proposed addendum to: guidelines on the quality, safety and efficacy of biotherapeutic protein products prepared by recombinant DNA technology. World Health Organization. http://www.who.int/biologicals/BS2251_WHO_RA_for_BTP_25_June_2015.pdf . Accessed 28 Aug 2015

Japan Ministry of Health Labour and Welfare (MHLW) (2009) Guidelines for the quality, safety and efficacy assurance of follow-on biologics [Yakushoku Shinsahatu 0304007 by MHLW]. Evaluation and Licensing Division, Pharmaceutical and Food Safety Bureau, Ministry of Health, Labour and Welfare. http://www.pmda.go.jp/files/000153851.pdf Accessed 28 July 2015

Ministry of Food and Drug Safety (MFDS) (2009) Guidelines on the evaluation of biosimilar products. Republic of Korea National Institute of Food and Drug Safety Evaluation. http://www.nifds.go.kr/en/research/bio.jsp . Accessed 28 July 2015

Health Sciences Authority, Health Products Regulation Group (2011) Guidance on registration of similar biological products in Singapore. Health Sciences Authority (HSA). http://www.hsa.gov.sg/content/dam/HSA/HPRG/Western_Medicine/Overview_Framework_Policies/Guidelines_on_Drug_Registration/Appendix%2017_Guidance%20on%20Registration%20of%20Similar%20Biological%20Products%20in%20Singapore%202011.pdf . Accessed 28 July 2015

Ministry of Health Malaysia, National Pharmaceutical Control Bureau (NPCB) (2008) Guidance document and guidelines for registration of biosimilars in Malaysia. Ministry of Health Malaysia. http://portal.bpfk.gov.my/index.cfm?menuid=90&q=biosimilar . Accessed 28 July 2015

Generics and Biosimilars Initiative (GaBI) (2012) India releases draft similar biologic guidelines. Pro Pharma Communications International. http://www.gabionline.net/Guidelines/India-releases-draft-similar-biologic-guidelines . Accessed 30 July 2015

Department of Biotechnology, Central Drugs Standard Control Organization (2012) Guidelines on similar biologics: regulatory requirements for marketing authorization in India. Government of India. http://dbtbiosafety.nic.in/Files%5CCDSCO-DBTSimilarBiologicsfinal.pdf . Accessed 30 July 2015

Generics and Biosimilars Initiative (GaBI) (2012) ‘Similar biologics’ approved and marketed in India. Pro Pharma Communications International. http://www.gabionline.net/Biosimilars/General/Similar-biologics-approved-and-marketed-in-India . Accessed 30 July 2015

Generics and Biosimilars Initiative (GaBI) (2014) China releases draft biosimilars guidance. Pro Pharma Communications International. http://www.gabionline.net/Guidelines/China-releases-draft-biosimilars-guidance . Accessed 25 July 2015

International Federation of Pharmaceutical Manufacturers and Associations (April 8-10, 2014) Biologic qualifiers: a global means to the identification and traceability of biotherapeutic medicines. Proceedings of the 58th Consultation on International Non-Proprietary Names for Pharmaceutical Substances. http://www.who.int/medicines/services/inn/58th_executive_summary.pdf . Accessed 30 July 2015

World Health Organization, Programme on International Nonproprietary Names (INN) (2015) Biological qualifier: an INN proposal. World Health Organization. http://www.who.int/medicines/services/inn/bq_innproposal201506.pdf.pdf . Accessed 30 July 2015

Traynor K (2014) Stakeholders discuss biosimilar naming, substitution. Am J Health Syst Pharm 71:446–447. doi: 10.2146/news140023

Bennett CL, Chen B, Hermanson T et al (2014) Regulatory and clinical considerations for biosimilar oncology drugs. Lancet Oncol 15:e594–e605. doi: 10.1016/S1470-2045(14)70365-1

Casadevall N, Edwards IR, Felix T, Graze PR, Litten JB, Strober BE, Warnock DG (2013) Pharmacovigilance and biosimilars: considerations, needs and challenges. Expert Opin Biol Ther 13:1039–1047. doi: 10.1517/14712598.2013.783560

The Pharmaceuticals and Medical Devices Agency Japan (2009) Guideline for the quality, safety, and effectiveness of biosimilar products. http://www.jpma.or.jp/ . Accessed 30 July 2015

Ministry of Health Labour and Welfare Pharmaceutical and Food Safety Bureau (2014) Handling of generic and trade name of biosimilars. Japan Ministry of Health. http://www.pmda.go.jp/files/000198125.pdf . Accessed 30 July 2015

Australian Government Department of Health, Therapeutic Goods Administration (2015) Naming conventions for biosimilars. Australian Government. https://www.tga.gov.au/book/naming-conventions-biosimilars . Accessed 29 July 2015

US Food and Drug Administration, Center for Drug Evaluation and Research (2015) Guidance for industry: nonproprietary naming of biological products (Draft). US Department of Health and Human Services, US Food and Drug Administration, Center for Drug Evaluation and Research (CDER), Center for Biologics Evaluation and Research (CBER). http://www.fda.gov/downloads/Drugs/GuidanceComplianceRegulatoryInformation/Guidances/UCM459987.pdf . Accessed 28 Aug 2015

Pineda C, Caballero-Uribe CV, de Oliveira MG, Lipszyc PS, Lopez JJ, Mataos Moreira MM, Azevedo VF (2015) Recommendations on how to ensure the safety and effectiveness of biosimilars in Latin America: a point of view. Clin Rheumatol 34:635–640. doi: 10.1007/s10067-015-2887-0

Vermeer NS, Straus SM, Mantel-Teeuwisse AK, Domergue F, Egberts TC, Leufkens HG, De Bruin ML (2013) Traceability of biopharmaceuticals in spontaneous reporting systems: a cross-sectional study in the FDA Adverse Event Reporting System (FAERS) and EudraVigilance databases. Drug Saf 36:617–625. doi: 10.1007/s40264-013-0073-3

Belton KJ (1997) Attitude survey of adverse drug-reaction reporting by health care professionals across the European Union. The European Pharmacovigilance Research Group. Eur J Clin Pharmacol 52:423–427

Bergvall T, Noren GN, Lindquist M (2014) vigiGrade: a tool to identify well-documented individual case reports and highlight systematic data quality issues. Drug Saf 37:65–77. doi: 10.1007/s40264-013-0131-x

World Health Organization (2015) The WHO programme for international drug monitoring. World Health Organization. http://www.who.int/medicines/areas/quality_safety/safety_efficacy/National_PV_Centres_Map/en/ . Accessed 30 July 2015

Hazell L, Shakir SA (2006) Under-reporting of adverse drug reactions: a systematic review. Drug Saf 29:385–396

Vermeer NS, Duijnhoven RG, Straus SM, Mantel-Teeuwisse AK, Arlett PR, Egberts AC, Leufkens HG, De Bruin ML (2014) Risk management plans as a tool for proactive pharmacovigilance: a cohort study of newly approved drugs in Europe. Clin Pharmacol Ther 96:723–731. doi: 10.1038/clpt.2014.184

Calvo B, Zuñiga L (2011) Risk management plan and pharmacovigilance system. Biopharmaceuticals: biosimilars. In: Nota G (ed) Risk management trends

Zuniga L, Calvo B (2010) Biosimilars: pharmacovigilance and risk management. Pharmacoepidemiol Drug Saf 19:661–669. doi: 10.1002/pds.1948

Rondon F, Bautista A, Salazar JC et al (2010) Etanar therapy in real-life patients with rheumatoid arthritis [abstract]. Arthritis Rheum 62:1811

Amgen (2015) Enbrel (etanercept) prescribing information. Amgen. http://pi.amgen.com/united_states/enbrel/derm/enbrel_pi.pdf . Accessed June 2015

Barile-Fabris LA, Irazoque-Palazuelos F, Hernández Vásquez R et al (2015) Incidence of adverse events in patients treated with intended copies of biologic therapeutic agents in Colombia and Mexico [abstract 1506]. Arthritis Rheum 66:S662. doi: 10.1007/s10067-014-2841-6

Uppsala Monitoring Centre, World Health Organization (2015) Reporting trends. http://who-umc.org/DynPage.aspx?id=108476&mn1=7347&mn2=7252&mn3=7322&mn4=7558 . Accessed 30 July 2015

Therapeutic Goods Administration (2011) Australian regulatory guidelines for biologicals (ARGB). Australian Government Department of Health. http://www.tga.gov.au/publication/australian-regulatory-guidelines-biologicals-argb . Accessed 4 Aug 2015

Scheinberg MA, Azevedo VF (2014) Biosimilars in rheumatology: perspective and concerns. Rheumatology (Oxford) 53:389–390. doi: 10.1093/rheumatology/ket210

Vital EM, Kay J, Emery P (2013) Rituximab biosimilars. Expert Opin Biol Ther 13:1049–1062. doi: 10.1517/14712598.2013.787064