Chapter 26. Discovery and Identification of Lead Compounds from Combinatorial Mixtures
Tài liệu tham khảo
Fenniri, 1996, Cur. Med. Chem., 3, 343, 10.2174/092986730305220302123912
Willard, 1996, Eur. J. Med. Chem., 31, 87, 10.1016/0223-5234(96)80441-7
Furka, 1995, Drug Dev. Res., 36, 1, 10.1002/ddr.430360102
Ecker, 1995, Biotechnology, 13, 351, 10.1038/nbt0495-351
Geysen, 1986, Mol. Immunol., 23, 709, 10.1016/0161-5890(86)90081-7
Oliphant, 1988, Nucl. Acids Res., 16, 7673, 10.1093/nar/16.15.7673
Furka, 1988, In. Abstr. 14th Int. Congr. Biochem. Prague, Czechoslovakia, 5, 47
Furka, 1991, Int. J. Protein Res, 37, 487, 10.1111/j.1399-3011.1991.tb00765.x
Houghten, 1993, Gene, 137, 7, 10.1016/0378-1119(93)90244-W
Burbaum, 1995, Proc. Natl. Acad. Sci. USA, 92, 6027, 10.1073/pnas.92.13.6027
Boutin, 1995, Trends in Pharm. Sci., 17, 8, 10.1016/0165-6147(96)81563-X
Chabala, 1995, Cur. Opin. Biotech., 6, 632, 10.1016/0958-1669(95)80104-9
Jayawickreme, 1994, Proc. Natl. Acad. Sci. USA, 91, 1614, 10.1073/pnas.91.5.1614
Quillan, 1995, Proc. Natl. Acad. Sci. USA, 92, 2894, 10.1073/pnas.92.7.2894
Salmon, 1996, Mol. Divers., 2, 57, 10.1007/BF01718701
Z. Yuan, “High Density Assay Formats for Screening Large Combinatorial Chemical Libraries”, Society for Biomolecular Screening 2nd Annual Conference, Basel, Switzerland, Oct. 14–17(1996)
N. H. Sigal, “New Screening Paradigms for the Evaluation of Small Molecule Combinatorial Libraries”, Second Annual High Throughput Screening for Drug Discovery Conference, San Diego, CA, June 14–16(1995)
Bock, 1992, Nature, 355, 564, 10.1038/355564a0
Tuerk, 1992, Proc. Natl. Acad. Sci. USA, 89, 6988, 10.1073/pnas.89.15.6988
Ellington, 1990, Nature, 346, 818, 10.1038/346818a0
Zuckermann, 1992, Proc. Natl. Acad. Sci. USA, 89, 4505, 10.1073/pnas.89.10.4505
B. A. Beutel, PCT patent WO95/27072(1995)
B. A. Beutel, “COMPILE: A Combinatorial Procedure for Indirect Ligand Eluciation”, Expoiting Molecular Diversity: Small Molecule Libraries For Drug Discovery, Cambridge Healthtech Institute Conference, La Jolla, CA Jan. 26–27(1995).
Evans, 1996, Nature Biotech., 14, 504, 10.1038/nbt0496-504
Fathi, 1996, J. Org. Chem., 61, 5600, 10.1021/jo960192+
Cheng, 1995, J. Am. Chem. Soc., 117, 8859, 10.1021/ja00139a023
Konings, 1996, J. Med Chem., 39, 2710, 10.1021/jm960168o
Wilson-Lingardo, 1996, J. Med. Chem., 39, 2720, 10.1021/jm960169g
Dooley, 1994, Science, 266, 2019, 10.1126/science.7801131
Loo, 1996, Annual Rep. In Med. Chem., 31, 319, 10.1016/S0065-7743(08)60471-6
Krchnak, 1995, Mol. Divers., 1, 193, 10.1007/BF01544958
Brummel, 1996, Anal. Chem., 68, 237, 10.1021/ac950998u
Haskins, 1995, Rapid Commun. Mass Sp., 9, 1437, 10.1002/rcm.1290091421
Sarkar, 1996, J. Am. Chem. Soc., 118, 2305, 10.1021/ja952434d
Yan, 1996, J. Org. Chem., 61, 7467, 10.1021/jo961416r
Brenner, 1992, Proc. Natl. Acad. Sci. USA, 89, 5381, 10.1073/pnas.89.12.5381
Needels, 1993, Proc. Natl. Acad. Sci. USA., 90, 10700, 10.1073/pnas.90.22.10700
Kerr, 1993, J. Am. Chem. Soc., 115, 2529, 10.1021/ja00059a070
Vagner, 1996, Proc. Natl. Acad. Sci. USA, 93, 8194, 10.1073/pnas.93.16.8194
Ohlmeyer, 1993, Proc. Natl. Acad. Sci. USA, 90, 10922, 10.1073/pnas.90.23.10922
Burbaum, 1995, Proc. Natl. Acad. Sci. USA, 92, 6027, 10.1073/pnas.92.13.6027
Ni, 1996, Methods in Enzymol., 267, 261, 10.1016/S0076-6879(96)67018-9
Ni, 1996, J. Med. Chem., 39, 1601, 10.1021/jm960043j
