Bioavailability study of fixed-dose tablet versus capsule formulation of amlodipine plus benazepril: A randomized, single-dose, two-sequence, two-period, open-label, crossover study in healthy volunteers

Current Therapeutic Research - Tập 66 - Trang 69-79 - 2005
Kuo-Liong Chien1,2, Chia-Lun Chao2, Ta-Cheng Su2
1Institute of Preventive Medicine, College of Public Health, National TaiwanUniversity, Taipei, Taiwan
2Department of Internal Medicine, National Taiwan University Hospital, Taipei, Taiwan

Tài liệu tham khảo

Guidelines Subcommittee, 1999, World Health Organization-International Society of Hypertension Guidelines for the Management of Hypertension. Guidelines Subcommittee, J Hypertens, 17, 151 Chobanian, 2003, The Seventh Report of the Joint National Committee on Prevention, Detection, Evaluation, and Treatment of High Blood Pressure, Hypertension, 42, 1206, 10.1161/01.HYP.0000107251.49515.c2 Lees, 1987, A clinical pharmacological study of nifedipine and lisinopril alone and in combination, J Cardiovasc Pharmacol., 10, S105, 10.1097/00005344-198706110-00038 Jakobsen, 1992, Unmasking of the hypotensive effect of nifedipine in normotensives by addition of the angiotensin converting enzyme inhibitor benazepril, J Hypertens, 10, 1045, 10.1097/00004872-199209000-00020 Brunel, 1991, Arterial and endocrine effects of a combination of an angiotensin converting enzyme inhibitor and a vasodilator in normotensive healthy volunteers, J Cardiovasc Pharmacol., 18, 175, 10.1097/00005344-199108000-00001 Meredith, 1992, Clinical pharmacokinetics of amlodipine, Clin Pharmacokinet., 22, 22, 10.2165/00003088-199222010-00003 Balfour, 1991, Benazepril. A review of its pharmacodynamic and pharmacokinetic properties, and therapeutic efficacy in hypertension and congestive heart failure, Drugs, 42, 511, 10.2165/00003495-199142030-00008 Fogari, 1997, Combined therapy with benazepril and amlodipine in the treatment of hypertension inadequately controlled by an ACE inhibitor alone, J Cardiovasc Pharmacol., 30, 497, 10.1097/00005344-199710000-00014 2000 Faulkner, 1986, The pharmacokinetics of amlodipine in healthy volunteers after single intravenous and oral doses and after 14 repeated oral doses given once daily, Br J Clin Pharmacol., 22, 21, 10.1111/j.1365-2125.1986.tb02874.x Sun, 1994, Pharmacokinetic interaction study between benazepril and amlodipine in healthy subjects, Eur J Clin Pharmacol., 47, 285, 10.1007/BF02570510 Kaiser, 1989, Pharmacokinetics of a new angiotensin-converting enzyme inhibitor, benazepril hydrochloride, in special populations, Am Heart J., 117, 746, 10.1016/0002-8703(89)90765-5 Williams, 1988, Amlodipine pharmacokinetics in healthy volunteers, J Clin Pharmacol., 28, 990, 10.1002/j.1552-4604.1988.tb03119.x Abernethy, 1992, Pharmacokinetics and pharmacodynamics of amlodipine, Cardiology, 80, 31, 10.1159/000175050 Kelly, 1990, Clinical pharmacokinetics of the newer ACE inhibitors. A review, Clin Pharmacokinet., 19, 177, 10.2165/00003088-199019030-00003 2000