Aromatic trivalent arsenicals: covalent yet reversible reagents for the agonist binding site of nicotinic receptors
Tài liệu tham khảo
Adamson, 1984, Inhibition of pyruvate dehydrogenase multienzyme complex from Escherichia coli with a radiolabeled bifunctional arsenoxide: evidence for an essential histidine residue at the active site of lipoamide dehydrogenase, Biochemistry, 23, 1269, 10.1021/bi00301a039
Bartels, 1970, Affinity oxidation of the reduced acetylcholine receptor, Biochim. Biophys. Acta, 203, 568, 10.1016/0005-2736(70)90193-8
Bertrand, 1990, Activation and blocking of neuronal nicotinic acetylchline receptor reconstituted in Xenopus oocytes, 87, 1993
Boyd, 1988, Expression and regulation of neuronal acetylcholine receptor mRNA in chick ciliary ganglia, Neuron, 1, 495, 10.1016/0896-6273(88)90180-8
Braswell, 1984, Pressure reversal of the action of octanol on postynaptic membranes from Torpedo, Br. J. Pharmacol., 83, 305, 10.1111/j.1476-5381.1984.tb10147.x
Brown, 1987, Spectroscopic characterization of thioredoxin covalently modified with monofunctional organoarsenical reagents, Biochemistry, 26, 863, 10.1021/bi00377a030
Czajkowski, 1991, Agonist binding site of Torpedo electric tissue nicotinic acetylcholine receptor, 266, 22603
Damle, 1978, Bromoacetylcholine as an affinity label of the acetylcholine receptor from Torpedo californica, Biophys. Res. Commun., 84, 845, 10.1016/0006-291X(78)91661-3
Dennis, 1988, Amino acids of the Torpedo marmorata acetycholine receptor α subunit labeled by a photoaffinity ligand for the acetylcholine binding site, Biochemistry, 27, 2346, 10.1021/bi00407a016
Ehrlich, 1909, Über den jetzigen Stand der Chemotherapie, Ber. dtsch. Chem. Ges., 42, 17, 10.1002/cber.19090420105
Frost, 1990, Uptake and binding of radiolabeled phenylarsine oxide in 3T3-L1 adipocytes, Biochem. J., 269, 589, 10.1042/bj2690589
Galzi, 1991, Functional architecture of the nicotinic acetylcholine receptor: from electric organ to brain, Annu. Rev. Pharmacol., 31, 37, 10.1146/annurev.pa.31.040191.000345
Heinemann, 1991, The nicotinic receptor genes, Clin. Neuropharmacol., 14S, s45, 10.1097/00002826-199114001-00007
Jauhiainen, 1988, Human plasma lecithin-cholesterol acyltransferase: the vicinal nature of cysteine 31 and cysteine 184 in the catalytic site, J. Biol. Chem., 263, 6525, 10.1016/S0021-9258(18)68673-9
Kao, 1986, Acetylcholine receptor binding site contains a disulfide crosslink between adjacent cystinyl residues, J. Biol. Chem., 261, 8085, 10.1016/S0021-9258(19)83877-2
Karlin, 1966, Effects of blocking sulfhydryl groups and of reducing disulfide bonds on the acetylcholine-activated permeability system of the electroplax, Biochim. Biophys. Acta, 126, 525, 10.1016/0926-6585(66)90010-0
Lindstrom, 1981, Production and assay of antibodies to acetylcholine receptors, Methods Enzymol., 74, 432, 10.1016/0076-6879(81)74031-X
Loring, 1990, Agmatine acts as an antagonist of neuronal nicotinic receptors, Br. J. Pharmacol., 99, 207, 10.1111/j.1476-5381.1990.tb14680.x
Loring, 1989, Characterization of nicotinic receptors in chick retina using a snake venom neurotoxin that blocks neuronal nicotinic receptor function, J. Neurosci., 9, 2423, 10.1523/JNEUROSCI.09-07-02423.1989
Loring, 1982, 125I-α-Bungarotoxin: effects of radiodecomposition on specific activity, J. Biol. Chem., 257, 1418, 10.1016/S0021-9258(19)68209-8
Loring, 1991, Ehrlich's magic bullet revisited: Aromatic arsenoxides as selective reagents for nicotinic receptors, Soc. Neurosci. Abstr., 17, 23
Loring, 1990, Pharmacological and biochemical properties of nicotinic receptors from chick retina, Eur. J. Neurosci., 2, 863, 10.1111/j.1460-9568.1990.tb00397.x
Leutje, 1991, Both α- and β-subunits contribute to the agonist sensitivity of neuronal nicotinic acetylcholine receptors, J. Neurosci., 11, 837, 10.1523/JNEUROSCI.11-03-00837.1991
Matter, 1990, Expression of neuronal nicotinic acetylcholine receptor genes in the developing chick visual system, EMBO J., 9, 1021, 10.1002/j.1460-2075.1990.tb08205.x
McLane, 1991, Structural determinants of alpha-bungarotoxin binding to the sequence 181–200 of the muscle nicotinic acetylcholine receptor alpha subunit: effects of cysteine/cystine modification, Biochemistry, 30, 4925, 10.1021/bi00234a013
Means, 1971, Chemical Modification of Proteins, 105
Pedersen, 1990, d-Tubocurarine binding sites are located at α-τ and α-δ subunit interfaces of the nicotinic acetylcholine receptor, 87, 2785
Ratnam, 1986, Structural heterogeneity of the α-subunits of the nicotinic acetylcholine receptor in relation to agonist affinity alkylation and antagonist binding, Biochemistry, 15, 4268, 10.1021/bi00363a014
Ravdin, 1979, Inhibition of neuronal acetylcholine sensitivity by alpha-toxins from Bungarus multicinctus venom, 76, 2072
Silman, 1969, Acetylcholine receptor: covalent attachment of depolarizing groups at the active site, Science, 164, 1420, 10.1126/science.164.3886.1420
Song, 1990, A binding site peptide fragment of the nicotinic acetylcholine receptor, 40, 63
Smythies, 1989, A possible structure for the nicotinic acetylcholine receptor, J. Receptor Res., 9, 199, 10.3109/10799898909066054
Stevenson, 1978, Inhibition of pyruvate dehydrogenase multienzyme complex from Eschericia coli with mono- and bifunctional arsenoxides, Biochemistry, 17, 2189, 10.1021/bi00604a026
Sussman, 1991, Atomic structure of acetylcholinesterase from Torpedo californica: a prototypic acetylcholine-binding protein, Science, 253, 872, 10.1126/science.1678899
Taylor, 1991, Distinctions in ligand binding sites on the nicotinic acetylcholine receptor, Ann. N.Y. Acad. Sci., 625, 568, 10.1111/j.1749-6632.1991.tb33893.x
Tzartos, 1981, Mapping of surface structures of Electrophorus acetycholine receptors using monoclonal antibodies, J. Biol. Chem., 256, 8635, 10.1016/S0021-9258(19)68891-5
Webb, 1966, Arsenicals, Vol. 3, 595
Whiting, 1991, Expression of nicotinic acetylcholine receptor subtypes in brain and retina, Mol. Brain Res., 10, 61, 10.1016/0169-328X(91)90057-5
