Antimicrobial activity of thiophene derivatives derived from ethyl (E)-5-(3-(dimethylamino)acryloyl)-4-methyl-2-(phenylamino)thiophene-3-carboxylate
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Riyadh S, Abdelhamid IA, Al-Matar HM, Hilmy NM, Elnagdi MH (2008) Enamines as precursors to polyfunctional heteroaromatic compounds; a decade of development. Heterocycles 75:1849–1905
Abu Shanab FA, Sherif SM, Mousa SA (2009) Dimethylformamide dimethyl acetal as a building block in heterocyclic synthesis. J Heterocycl Chem 46:801–872
Shawali AS (2012) Bis-Enaminones as versatile precursors for terheterocycles: synthesis and reactions. ARKIVOC 1:383–431
Wang F, Jin L, Kong L, Li X (2017) Cobalt(III)- and rhodium(III)-catalyzed C–H amidation and synthesis of 4-quinolones: C–H activation assisted by weakly coordinating and functionalizable enaminone. Org Lett 19(7):1812–1815
Mabkhot YN, Kaal NA, Alterary S, Al-Showiman SS, Barakat A, Ghabbour HA, Frey W (2015) Synthesis, in-vitro antibacterial, antifungal, and molecular modeling of potent anti-microbial agents with a combined pyrazole and thiophene pharmacophore. Molecules 20:8712–8729
Sakamaki S, Kawanishi E, Koga Y, Yamamoto Y, Kuriyama C, Matsushita Y, Ueta K, Nomura S (2013) Synthesis and biological evaluation of thiophene-C-glucosides as sodium-dependent glucose cotransporter 2 inhibitors. Chem Pharm Bull 61(10):1037–1043
Chaudhary A, Jha KK, Kumar S (2012) Biological diversity of thiophene: a review. J Adv Sci Res 3(3):03–10
Ansary AK, Omar HA (2001) Synthesis and anti -in fl amatory activity of some thieno [2,3d] pyrimidmone derivatives. Bull Fac Pharm 39:17
Lepifre FF, Lena GR, Autier V, Kergoat M, Faveriel LR, Charon CG, Raynal SN, Audet AM (2015) Useful thiophene derivatives in the treatment of diabetes. United States patent application 20150197530
Mongevega A, Aldama I, Robbani MM, Fernandez E (1980) The synthesis of 11H-1,2,4-triazolo [4,3-b] pyridazino [4,5-b] indoles, 11H-tetrazolo [4,5-b] pyridazino [4,5-b] indoles and 1,2,4-triazolo [3,4-f]-1,2,4-triazino [4,5-a]i ndoles. J Heterocycl Chem 17:77–80
Mabkhot YN, Alatibi F, El-Sayed NNE, Kheder NA, Al-Showiman SS (2016) Synthesis and structure-activity relationship of some new thiophene-based heterocycles as potential antimicrobial agents. Molecules 21(8):1036
Chen HJ, Wang Wl, Wang GF, Shi LP, Gu M, Ren YD, Hou LF (2008) Rational design and synthesis of 2,2-bisheterocycle tandem derivatives as non-nucleoside hepatitis B virus inhibitors. Med Chem 3:1316–1321
Gotteland JP, Planty B, Junquero D, Delhon A, Halazy S (1998) Sulfonamide derivatives of benzylamine block cholesterol biosynthesis in HepG2 cells: a new type of potent squalene epoxidase inhibitors. Bioorg Med Chem Lett 8:1337–1342
Hassan NA, Shawali AS, Abu-Zied KM, Osman DA (2013) Synthesis and antiviral evaluation of some new thieno[2,3-d]pyrimidine S-glycosides. J Appl Sci Res 9(1):833–842
Valderrama JA, Espinoza O, Rodriguez J, Theoduloz C (2009) Synthesis and antitumor evaluation of thiophene analogs of kigelinone. Lett Org Chem 6:278–281
Hassaneen H, Eid E, Eid H, Farghaly TA, Mabkhot Y (2017) Facial regioselective synthesis of novel bioactive spiropyrrolidine/pyrrolizine-oxindole derivatives via a three components reactions as potential antimicrobial agents. Molecules 22(3):357–371
Dawood DH, Batran RZ, Farghaly TA, Khedr MA, Abdulla MM (2015) New coumarin derivatives as potent selective COX-2 inhibitors; synthesis, anti-inflammatory, QSAR and molecular modeling studies. Arch Pharm Chem Life Sci 348:875–888
Farghaly TA, Abdallah MA, Masaret GS, Muhammad ZA (2015) New and efficient approach for synthesis of novel bioactive [1,3,4]thiadiazoles incorporated with 1,3-thiazole moiety. Eur J Med Chem 97:320–333
Farghaly TA, Hassaneen HME, Elzahabi HAS (2015) Eco-friendly synthesis and 2D-QSAR study of novel pyrazolinesas potential anticolon cancer agents. Med Chem Res 24:652–668
Awad HM, Fayad W, El-Hallouty SM, Farghaly TA, Abdallah MM (2016) Anticancer activity of some [1, 2, 4] triazepino[2,3-a] quinazoline derivatives: monolayer and multicellular spheroids in vitro models. Med Chem Res 25(9):1952–1957
Farghaly TA, Abdallah MA, Muhammad ZA (2016) 2,7-Diarylidene-cycloheptanone, hydrazonoyl chlorides and heterocyclic amines as precursors for synthesis of bioactive new fused cycloheptapyrimidine derivatives. Curr Org Syn 13(2):291–299
Al Majid AMA, Barakat A, Mabkhot YN, Al-Agamy MHM (2016) Synthesis, and characterization of a new series of sulfite and sulfate derivatives of D-Mannitol. J Saudi Chem Soc 20:307–312
Tighadouni S, Radi S, Sirajuddin M, Akkurt M, Özdemir N, Ahmad M, Mabkhot YN, Ben Hadda T (2016) In vitro antifungal, anticancer activities and POM analyses of a novel bioactive schiff base 4-{[(E)-furan-2-ylmethylidene]amino}p-henol: synthesis, characterization and crystal structure. J Chem Soc Pak 38:157–165
Farghaly TA, Abdallah MA, Mahmoud HK (2015) Synthesis of novel 1,2,4-triazoles and triazolo-thiadiazines as anticancer agents. Turk J Chem 39:955–969
Mabkhot YN, Kaal NA, Alterary S, Al-Showiman SS, Barakat A, Ghabbour HA, Frey W (2015) Synthesis, in-vitro antibacterial, antifungal, and molecular modeling of potent anti-microbial agents with a combined pyrazole and thiophene pharmacophore. Molecules 20:8712–8729
Elassar AA, El-Khair AA (2003) Recent developments in the chemistry of enaminones. Tetrahedron 59:8463–8480
Mabkhot YN, Barakat A, Al-Majid AM, AlShahrani SA (2012) Comprehensive and facile synthesis of some functionalized bis-heterocyclic compounds containing a thieno[2,3-b]thiophene Motif. Int J Mol Sci 13:2263–2275
Riyadh SM (2011) Enaminones as building blocks for the synthesis of substituted pyrazoles with antitumor and antimicrobial activities. Molecules 16:1834–1853
Cruickshank R, Duguid JP, Marion BP, Swain RH (1975) A medicinal microbiology, vol 2, 12th edn. Churchill Livingstone, London, pp 196–202