Analgesic and other pharmacological activities of an enkephalin analogue, syndyphalin (SD)-25

European Journal of Pharmacology - Tập 85 - Trang 133-142 - 1982
Hideo Nakamura1, Yoshiaki Kiso2, Satoru Motoyoshi1, Naoyuki Yoshida1, Katsumi Ishii1, Yuichi Yokoyama1, Toshiaki Kadokawa1, Masanao Shimizu1
1Department of Pharmacology, Research Laboratories, Dainippon Pharmaceutical Co., Ltd. Suita, Osaka, 564 Japan
2Faculty of Pharmaceutical Sciences, University of Tokushima, Tokushima 770, Japan

Tài liệu tham khảo

Bass, 1965, Effect of ligation and morphine on electric and motor activity of dog duodenum, Am. J. Physiol., 208, 908, 10.1152/ajplegacy.1965.208.5.908 Bellet, 1980, Central cardiovascular effects of narcotic analgesics and enkephalins in rats, Br. J. Pharmacol., 71, 365, 10.1111/j.1476-5381.1980.tb10949.x Belluzzi, 1976, Analgesia induced in vivo by central administration of enkephalin in rat, Nature, 260, 625, 10.1038/260625a0 Bhargava, 1977, Opiate-like action of methionine-enkephalin in inhibiting morphine abstinence syndrome, European J. Pharmacol., 41, 81, 10.1016/0014-2999(77)90375-2 Bhargava, 1978, New in vivo evidence for narcotic agonistic property of leucine-enkephalin, J. Pharm. Sci., 67, 136, 10.1002/jps.2600670141 Bolme, 1978, Cardiovascular effects of morphine and opioid peptides following intracisternal administration in chloralose-anesthetized rats, European J. Pharmacol., 48, 319, 10.1016/0014-2999(78)90090-0 Brady, 1981, Effects of intraventricular morphine and enkephalins on locomotor activity in nondependent, morphine-dependent and postdependent rats, J. Pharmacol. Exp. Ther., 218, 613 Buckett, 1964, A new test for morphine-like physical dependence (addiction liability) in rats, Psychopharmacology, 6, 410, 10.1007/BF00429568 Buescher, 1976, Evidence for analgesic activity of enkephalin in the mouse, Nature, 261, 423, 10.1038/261423a0 Chapman, 1980, Methionine-enkephalin antagonism and endorphin potentiation of narcotic-induced analgesia, European J. Pharmacol., 65, 369, 10.1016/0014-2999(80)90341-6 Denavit-Saubie, 1978, Effects of opiates and methionine-enkephalin on pontine and bulbar respiratory neurons of the cat, Brain Res., 155, 55, 10.1016/0006-8993(78)90305-0 Dupont, 1977, Extremely rapid degradation of [3H]-methionine-enkephalin by various rat tissues in vivo and in vitro, Life Sci., 21, 907, 10.1016/0024-3205(77)90254-5 Dutta, 1977, Enkephalin analogues eliciting analgesia after intravenous injection, Life Sci., 21, 559, 10.1016/0024-3205(77)90097-2 Feinberg, 1976, The opiate receptor: A model explaining structure-activity relationships of opiate agonists and antagonists, 73, 4215 Feldberg, 1978, Central cardiovascular effects of enkephalins and C-fragment of lipoprotein, J. Physiol. (London), 280, 18p Flórez, 1980, Respiratory effects of β-endorphin, D-ala2-met-enkephalinamide, and met-enkephalin injected into the lateral ventricule and the pontomedullary subarachnoid space, Brain Res., 199, 197, 10.1016/0006-8993(80)90240-1 Green, 1953, Analgesic and other properties of 3,3-dithienylalkenylamines, Br. J. Pharmacol., 8, 2 Haffner, 1929, Experimentelle Pruefung Schmerzstillender Mittel, Dtsch. Med. Wochensch., 55, 731, 10.1055/s-0028-1126487 Janssen, 1957, A new series of potent analgesics: Dextro 2:2-diphenyl-3-methyl-4-morpholinobutyrylprolidine and related amides. Part I. Chemical structure and pharmacological activity, J. Pharm. Pharmacol., 9, 381, 10.1111/j.2042-7158.1957.tb12290.x Kiso, 1981, Super-active enkephalin analogues. Simple tripeptide hydroxyalkylamides exhibit surprisingly high and long-lasting opioid activities, Naturwissenschaften, 68, 210, 10.1007/BF01047210 Kokka, 1965, Some effects of morphine on respiration and metabolism of rats, J. Pharmacol. Exp. Ther., 148, 386 Konturek, 1980, Influence of methionine-enkephalin and morphine on myoelectric activity of small bowel, Am. J. Physiol., 238, G384 Laubie, 1977, Central cardiovascular effects of morphinomimetic peptides in dogs, European J. Pharmacol., 46, 67, 10.1016/0014-2999(77)90146-7 Litchfield, 1949, A simplified method of evaluating dose-effect experiments, J. Pharmacol. Exp. Ther., 96, 99 Lord, 1977, Endogenous opioid peptides: multiple agonists and receptors, Nature, 267, 495, 10.1038/267495a0 Luján, 1981, Pharmacological characterization of opiate physical dependence in the isolated ileum of the guinea-pig, Br. J. Pharmacol., 73, 859, 10.1111/j.1476-5381.1981.tb08739.x Martin, 1976, The effects of morphine and nalorphine-like drugs in the non-dependent and morphine-dependent chronic spinal dog, J. Pharmacol. Exp. Ther., 197, 517 Martin, 1962, Interactions between nalorphine and morphine in the decerebrate cat, J. Pharmacol. Exp. Ther., 138, 113 Martin, 1963, Tolerance to and physical dependence on morphine in rats, Psychopharmacology, 4, 247, 10.1007/BF00408180 Morley, 1980, Structure-activity relationships of enkephalin-like peptides, Ann. Rev. Pharmacol. Toxicol., 20, 81, 10.1146/annurev.pa.20.040180.000501 Nakamura, 1978, Some altered responses in rats formerly dependent on morphine, Psychopharmacology, 56, 269, 10.1007/BF00432849 Nakamura, 1975, A substitution test for morphine-like physical dependence in morphine-dependent rats, Folia Pharmacol. Japon., 71, 105p Nakamura, 1976, Comparative study of 1-cyclohexyl-4-(1,2-diphenylethyl)-piperazine and its enantiomorphs on analgesic and other pharmacological activities in experimental animals, Arch. Int. Pharmacodyn., 221, 105 Nakamura, 1977, Effect of morphine and methamphetamine on spontaneous locomotor activity in grouped mice, Jap. J. Pharmacol., 27, 50p, 10.1016/S0021-5198(19)66411-5 Nakamura, 1977, Effects of abuse drugs on spontaneous locomotor activity in grouped mice, 11 Nakamura, 1973, Further studies on the mouse jumping test as a screening method to estimate the physical dependence capacity of analgesics, Folia Pharmacol. Japon., 69, 326p Oka, 1980, Enkephalin receptor in the rabbit ileum, Br. J. Pharmacol., 68, 193, 10.1111/j.1476-5381.1980.tb10406.x Oka, 1981, Enkephalin (opiate) receptors in the intestine, Trends Pharmacol. Sci., 12, 328, 10.1016/0165-6147(81)90356-4 Saelens, 1971, The mouse jumping test - a simple screening method to estimate the physical dependence capacity of analgesics, Arch. Int. Pharmacodyn., 190, 213 Simon, 1978, Effect of enkephalins on arterial blood pressure are reduced by propranolol, Clin. Sci. Mol. Med., 55, 237s Stewart, 1978, Central and peripheral actions of morphine on intestinal transit, J. Pharmacol. Exp. Ther., 205, 547 Tortella, 1980, D-Ala2-methionine-enkephalinamide self-administration in the morphine-dependent rat, Psychopharmacology, 69, 143, 10.1007/BF00427640 Vaught, 1978, Characterization of leucine and methionine-enkephalin and their interaction with morphine on the guinea pig ileal longitudinal muscle, Res. Commun. Chem. Pathol. Pharmacol., 21, 391 Vaught, 1979, Differential effects of leucine and methionine enkephalin on morphine-induced analgesia, acute tolerance and dependence, J. Pharmacol. Exp. Ther., 208, 86 Waterfield, 1977, In vitro pharmacology of the opioid peptides, enkephalins and endorphins, European J. Pharmacol., 43, 107, 10.1016/0014-2999(77)90123-6 Wei, 1981, Enkephalin analogs and physical dependence, J. Pharmacol. Exp. Ther., 216, 12 Wüster, 1980, The direction of opioid agonists towards μ, δ- and ϵ-receptors in the vas deferens of the mouse and the rat, Life Sci., 27, 163, 10.1016/0024-3205(80)90459-2 Zobrist, 1981, Characterization of the respiratory activity of (D-ala2)methionine-enkephalinamide, European J. Pharmacol., 70, 121, 10.1016/0014-2999(81)90206-5