A semi-automated method for measuring the potential for protein covalent binding in drug discovery

S.H. Day1, A. Mao2, R. White3, T. Schulz-Utermoehl4, R. Miller2, M.G. Beconi2
1Medicinal Chemistry, Merck Frosst Centre for Therapeutic Research, Merck Frosst Canada and Co., 16711 Trans Canada Hwy., Kirkland, Quebec, Canada H9H 3L1
2Drug Metabolism, Merck and Co., Inc., Rahway, NJ, USA
3Drug Metabolism, Merck and Co., Inc., West Point, PA, USA
4Medicinal Chemistry, Drug Metabolism Section, Merck Sharp and Dohme, Terlings Park, Harlow, Essex, United Kingdom

Tài liệu tham khảo

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