A public-private partnership to unlock the untargeted kinome

Nature Chemical Biology - Tập 9 Số 1 - Trang 3-6 - 2013
Stefan Knapp1, Paulo Arruda2, Patrick Münzer3, S.K. Burley4, David H. Drewry5, A.M. Edwards6, Doriano Fabbro7, Stefan Laufer8, Nathanael S. Gray9, Bernhard Küster10, Karen Lackey8, Paulo Mazzafera2, Nicholas C. O. Tomkinson11, Timothy M. Willson12, Robert N. Young3, William J. Zuercher12
1Department of Clinical Pharmacology, University of Oxford, Oxford, UK
2Universidade Estadual de Campinas
3Institute of Cancer Research
4University of california at San Diego
5(GlaxoSmithKline)
6STRUCTURAL GENOMICS CONSORTIUM
7#N##TAB##TAB##TAB##TAB# Novartis#N##TAB##TAB##TAB#
8Hoffmann- La Roche
9Harvard University
10Technical University of Munich
11University of Strathclyde
12Timothy M. Willson and William J. Zuercher are in the Department of Chemical Biology at GlaxoSmithKline, David H. Drewry, Research Triangle Park, North Carolina, USA.,

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Tài liệu tham khảo

Fedorov, O., Muller, S. & Knapp, S. Nat. Chem. Biol. 6, 166–169 (2010).

Edwards, A.M. et al. Nature 470, 163–165 (2011).

Bantscheff, M. et al. Nat. Biotechnol. 25, 1035–1044 (2007).

Patricelli, M.P. et al. Chem. Biol. 18, 699–710 (2011).

Davis, M.I. et al. Nat. Biotechnol. 29, 1046–1051 (2011).

Lin, X. et al. J. Med. Chem. 55, 5749–5759 (2012).

Fedorov, O. et al. Proc. Natl. Acad. Sci. USA 104, 20523–20528 (2007).

Frye, S.V. Nat. Chem. Biol. 6, 159–161 (2010).

Workman, P. & Collins, I. Chem. Biol. 17, 561–577 (2010).

Weigelt, J. EMBO Rep. 10, 941–945 (2009).

Cohen, P. Biochem. J. 425, 53–54 (2010).

Dowling, J.E. et al. ACS Med. Chem. Lett. 3, 278–283 (2012).

Al-Lazikani, B., Banerji, U. & Workman, P. Nat. Biotechnol. 30, 679–692 (2012).

Di Paolo, J.A. et al. Nat. Chem. Biol. 7, 41–50 (2011).

Deng, X. et al. Nat. Chem. Biol. 7, 203–205 (2011).

Medina, J.R. et al. J. Med. Chem. 54, 1871–1895 (2011).

Zhang, T. et al. Chem. Biol. 19, 140–154 (2012).

Zhang, J. et al. Natur. 463, 501–506 (2010).

Fedorov, O. et al. Chem. Biol. 18, 67–76 (2011).

Mott, B.T. et al. Bioorg. Med. Chem. Lett. 19, 6700–6705 (2009).

Shimomura, T. et al. Mol. Cancer Ther. 9, 157–166 (2010).

Koeberle, S.C. et al. Nat. Chem. Biol. 8, 141–143 (2011).

Bergamini, G. et al. Nat. Chem. Biol. 8, 576–582 (2012); corrigendum 8, 737 (2012).

Golding, S.E. et al. Mol. Cancer Ther. 8, 2894–2902 (2009).