A liposomal fluorescence assay to study permeation kinetics of drug-like weak bases across the lipid bilayer

Journal of Controlled Release - Tập 173 - Trang 102-109 - 2014
Klaus Eyer1, Franziska Paech2, Friedrich Schuler1, Phillip Kuhn1, Reinhard Kissner3, Sara Belli2, Petra S. Dittrich1, Stefanie D. Krämer2
1Bioanalytics, Laboratory of Organic Chemistry, Department of Chemistry and Applied Biosciences, ETH Zurich, Wolfgang-Pauli-Strasse 10, CH-8093 Zürich, Switzerland
2Biopharmacy and Radiopharmaceutical Sciences, Institute of Pharmaceutical Sciences, Department of Chemistry and Applied Biosciences, ETH Zurich, Wolfgang-Pauli-Strasse 10, CH-8093 Zürich, Switzerland
3Bioinorganic and Solution Chemistry, Laboratory of Inorganic Chemistry, Department of Chemistry and Applied Biosciences, ETH Zurich, Wolfgang-Pauli-Strasse 10, CH-8093 Zürich, Switzerland

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