Discovery of the antidepressant and anti-emetic efficacy of substance P receptor (NK1) antagonists

Trends in Pharmacological Sciences - Tập 20 - Trang 485-490 - 1999
Nadia M.J Rupniak1, Mark S Kramer2,3
1Merck Sharp & Dohme Neuroscience Research Centre, Harlow, Essex, UK CM20 2QR
2Clinical Neuroscience, Merck Research Laboratories, West Point, Philadelphia, PA 19456, USA
3Thomas Jefferson Medical College, Department of Psychiatry and Human Behavior, Philadelphia, PA 19107, USA

Tài liệu tham khảo

Kramer, 1998, Science, 281, 1640, 10.1126/science.281.5383.1640 Quartara, 1998, Neuropeptides, 32, 1, 10.1016/S0143-4179(98)90015-4 Snider, 1991, Science, 251, 435, 10.1126/science.1703323 Beresford, 1991, Br. J. Pharmacol., 104, 292, 10.1111/j.1476-5381.1991.tb12423.x Rupniak, 1997, Eur. J. Pharmacol., 326, 201, 10.1016/S0014-2999(97)85415-5 Rupniak, 1993, Br. J. Pharmacol., 110, 1607, 10.1111/j.1476-5381.1993.tb14008.x Rupniak, 1999, 135 Lembeck, 1953, Arch. Exp. Path. Pharmacol., 219, 197 Chang, 1971, Nature New Biol., 232, 86, 10.1038/232343a0 Henry, 1976, Brain Res., 114, 439, 10.1016/0006-8993(76)90965-3 Hokfelt, 1975, Brain Res., 100, 235, 10.1016/0006-8993(75)90481-3 Duggan, 1987, Brain Res., 403, 345, 10.1016/0006-8993(87)90073-4 Shults, 1984, Peptides, 5, 1097, 10.1016/0196-9781(84)90177-3 de Koninck, 1991, Proc. Natl. Acad. Sci. U. S. A., 88, 11344, 10.1073/pnas.88.24.11344 Block, 1998, Neurology, 50, A225 Kramer, 1995, Biol. Psychiatry, 37, 462, 10.1016/0006-3223(94)00190-E Armstrong, 1981, J. Comp. Neurol., 196, 505, 10.1002/cne.901960312 Andrews, 1994, 255 Matsumoto, 1999, Gan To Kagaku Ryoho, 26, 535 Tattersall, 1994, Neuropharmacology, 33, 259, 10.1016/0028-3908(94)90018-3 Tattersall, 1996, Neuropharmacology, 35, 1121, 10.1016/S0028-3908(96)00020-2 Rudd, 1996, Br. J. Pharmacol., 119, 931, 10.1111/j.1476-5381.1996.tb15761.x Kris, 1997, J. Natl. Cancer Inst., 89, 817, 10.1093/jnci/89.11.817 Hesketh, 1999, J. Clin. Oncol., 17, 338, 10.1200/JCO.1999.17.1.338 Navari, 1999, New Engl. J. Med., 340, 190, 10.1056/NEJM199901213400304 Tamiya, 1990, Neurosci. Lett., 110, 11, 10.1016/0304-3940(90)90779-9 Elliott, 1991, Neuropeptides, 19, 119, 10.1016/0143-4179(91)90141-5 Elliott, 1992, Behav. Brain Res., 51, 77, 10.1016/S0166-4328(05)80314-6 Elliott, 1986, Brain Res., 385, 379, 10.1016/0006-8993(86)91087-5 Minabe, 1996, Synapse, 22, 35, 10.1002/(SICI)1098-2396(199601)22:1<35::AID-SYN4>3.0.CO;2-J Seabrook, 1995, Eur. J. Pharmacol., 273, 113, 10.1016/0014-2999(94)00681-V Whitty, 1997, J. Comp. Neurol., 382, 394, 10.1002/(SICI)1096-9861(19970609)382:3<394::AID-CNE6>3.0.CO;2-Z Shibata, 1990, J. Pharmacol. Exp. Ther., 255, 388 Miller, 1996, Biol. Psychiatry, 39, 911, 10.1016/0006-3223(95)00098-4 Gabbard, 1995, 465 Mantyh, 1984, Brain Res., 307, 147, 10.1016/0006-8993(84)90470-0 Baker, 1991, Neuroscience, 42, 757, 10.1016/0306-4522(91)90043-N Elliott, 1988, Exp. Brain Res., 381, 354 Aguiar, 1996, Physiol. Behav., 60, 1183, 10.1016/0031-9384(96)00156-4 Krase, 1994, Behav. Brain Res., 63, 81, 10.1016/0166-4328(94)90053-1 Culman, 1995, Can. J. Physiol. Pharmacol., 73, 885, 10.1139/y95-122 Brodin, 1994, Neuropeptides, 26, 253, 10.1016/0143-4179(94)90079-5 Siegel, 1984, Neurochem. Int., 6, 783, 10.1016/0197-0186(84)90011-1 Shirayama, 1996, Brain Res., 739, 70, 10.1016/S0006-8993(96)00812-8 Berrettini, 1985, Biol. Psychiatry, 20, 965, 10.1016/0006-3223(85)90193-3 Bannon, 1986, Nature, 306, 791, 10.1038/306791a0 Barton, 1999, Br. J. Pharmacol., 126, 284P Hahn, 1999, Neuroscience Zernig, 1992, Neurosci. Lett., 143, 169, 10.1016/0304-3940(92)90258-9 File, 1997, Pharmacol. Biochem. Behav., 58, 747, 10.1016/S0091-3057(97)90002-2 Shaikh, 1993, Brain Res., 625, 283, 10.1016/0006-8993(93)91070-9 Dubinsky, 1971, Neuropharmacology, 10, 537, 10.1016/0028-3908(71)90019-0 Williams, 1998, Inv. Drugs, 1, 887