T-226296: a novel, orally active and selective melanin-concentrating hormone receptor antagonist

European Journal of Pharmacology - Tập 438 - Trang 129-135 - 2002
Shiro Takekawa1, Asano Asami1, Yuji Ishihara2, Jun Terauchi2, Kaneyoshi Kato2, Yukio Shimomura1, Masaaki Mori1, Hitomi Murakoshi3, Koki Kato3, Nobuhiro Suzuki1, Osamu Nishimura1, Masahiko Fujino1
1Discovery Research Laboratories I, Pharmaceutical Research Division, Takeda Chemical Industries, Ltd., Wadai 10, Tsukuba, Ibaraki 300-4293, Japan
2Medicinal Chemistry Research Laboratories II, Osaka 532-8686, Japan
3Pharmaceutical Research Laboratories II, Osaka 532-8686, Japan

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