ECE-1: A membrane-bound metalloprotease that catalyzes the proteolytic activation of big endothelin-1
Tóm tắt
Từ khóa
Tài liệu tham khảo
Ahn, 1992, The endothelin-converting enzyme from human umbilical vein is a membrane-bound metalloprotease similar to that from bovine aortic endothelial cells, 89, 8606
Arai, 1990, Cloning and expression of a cDNA encoding an endothelin receptor, Nature, 348, 730, 10.1038/348730a0
Benigni, 1993, A specific endothelin subtype A receptor antagonist protects against injury in renal disease progression, Kidney Int., 44, 440, 10.1038/ki.1993.263
Bloom, 1993, Acute cyclosporine-induced renal vasoconstriction is mediated by endothelin-1, Surgery, 114, 480
Chen, 1987, High-efficiency transformation of mammalian cells by plasmid DNA, Mol. Cell. Biol., 7, 2745, 10.1128/MCB.7.8.2745
Clozel, 1993, Pathophysiological role of endothelin revealed by the first orally active endothelin receptor antagonist, Nature, 365, 759, 10.1038/365759a0
Fernandez, 1992, Internal protein sequence analysis: enzymatic digestion for less than 10 μg of protein bound to polyvinylidene difluoride or nitrocellulose membranes, Anal. Biochem., 201, 255, 10.1016/0003-2697(92)90336-6
Gellai, 1994, Reversal of postischemic acute renal failure with a selective endothelinA receptor antagonist in the rat, J. Clin. Invest., 93, 900, 10.1172/JCI117046
Giaid, 1991, Topographical localisation of endothelin mRNA and peptide immunoreactivity in neurons of the human brain, Histochemistry, 95, 303, 10.1007/BF00266781
Giaid, 1993, Expression of endothelin-1 in lungs of patients with pulmonary hypertension, N. Engl. J. Med., 328, 1732, 10.1056/NEJM199306173282402
Grover, 1993, The endothelin-1 receptor antagonist BQ-123 reduces infarct size in a canine model of coronary occlusion and reperfusion, Cardiovasc. Res., 27, 1613, 10.1093/cvr/27.9.1613
Imai, 1992, Concomitant expression of receptor subtype and isopeptide of endothelin by human adrenal gland, Biochem. Biophys. Res. Commun., 182, 1115, 10.1016/0006-291X(92)91847-J
Inoue, 1989, The human endothelin family: three structurally and pharmacologically distinct isopeptides predicted by three separate genes, 86, 2863
Inoue, 1989, The human preproendothelin-1 gene, J. Biol. Chem., 264, 14954, 10.1016/S0021-9258(18)63795-0
Ito, 1993, Endothelin-1 is an autocrine/paracrine factor in the mechanism of angiotensin II-induced hypertrophy in cultured rat cardiomyocytes, J. Clin. Invest., 92, 398, 10.1172/JCI116579
Itoh, 1993, A novel endothelin ETA receptor antagonist, BQ-485, and its preventive effect on experimental cerebral vasospasm in dogs, Biochem. Biophys. Res. Commun., 195, 969, 10.1006/bbrc.1993.2139
Kivlighn, 1993, Effects of BQ-123 on renal function and acute cyclosporine-induced renal dysfunction, Kidney Int., 45, 131, 10.1038/ki.1994.15
Kurihara, 1994, Elevated blood pressure and craniofacial abnormalities in mice deficient in endothelin-1, Nature, 368, 703, 10.1038/368703a0
Lee, 1991, Cloning of the GATA-binding protein that regulates endothelin-1 gene expression in endothelial cells, J. Biol. Chem., 266, 16188, 10.1016/S0021-9258(18)98533-9
Lee, 1991, Molecular cloning and primary structure of Kell blood group protein, 88, 6353
Malfroy, 1988, Molecular cloning and amino acid sequence of human enkephalinase (neutral endopeptidase), FEBS Lett., 229, 206, 10.1016/0014-5793(88)80828-7
McMahon, 1991, Phosphoramidon blocks the pressor activity of porcine big endothelin-1(139) in vivo and conversion of big endothelin-1(139) to endothelin-1(121) in vitro, 88, 703
Nakajima, 1989, Synthesis of endothelin-1 analogues, endothelin-3, and sarafotoxin S6b: structure-activity relationships, J. Cardiovasc. Pharmacol., 13, S8, 10.1097/00005344-198900135-00004
Nishikibe, 1993, Antihypertensive effect of a newly synthesized endothelin antagonist, BQ-123, in a genetic hypertensive model, Life Sci., 52, 717, 10.1016/0024-3205(93)90233-S
Nishikori, 1991, Receptor binding affinity and biological activity of C-terminal elongated forms of endothelin-1, Neurochem. Int., 18, 535, 10.1016/0197-0186(91)90152-4
Ohlstein, 1994, SB 209670, a rationally designed potent nonpeptide endothelin receptor antagonist
Ohnaka, 1993, Purification and characterization of a phosphoramidonsensitive endothelin-converting enzyme in porcine aortic endothelium, J. Biol. Chem., 268, 26759, 10.1016/S0021-9258(19)74378-6
Okada, 1993, Big endothelin-1 structure important for specific processing by endothelin-converting enzyme of bovine endothelial cells, Eur. J. Biochem., 218, 493, 10.1111/j.1432-1033.1993.tb18401.x
Roques, 1993, Neutral endopeptidase 24.11: structure, inhibition, and experimental and clinical pharmacology, Pharmacol. Rev., 45, 87
Rosolowsky, 1994, Endothelial cells stimulate aldosterone release from bovine adrenal zona glomerulosa cells, Am. J. Physiol., 266, 107
Sakamoto, 1993, Distinct subdomains of human endothelin receptors determine their selectivity to ETA-selective antagonist and ETB-selective agaonists, J. Biol. Chem., 268, 8547, 10.1016/S0021-9258(18)52910-0
Sakurai, 1990, Cloning of a cDNA encoding a non-isopeptide-selective subtype of the endothelin receptor, Nature, 348, 732, 10.1038/348732a0
Sawamura, 1991, Phosphoramidon inhibits the intracellular conversion of big endothelin-1 to endothelin-1 in cultured endothelial cells, Biochem. Biophys. Res. Commun., 174, 779, 10.1016/0006-291X(91)91485-U
Seidah, 1993, Mammalian paired basic amino acid convertases of prohormones and proproteins, Ann. N Y Acad. Sci., 680, 135, 10.1111/j.1749-6632.1993.tb19680.x
Sogabe, 1993, Pharmacological profile of FR139317, a novel, potent endothelin ETA receptor antagonist, J. Pharmacol. Exp. Ther., 264, 1040
Stein, 1994, The discovery of sulfonamide endothelin antagonists and the development of the orally active ETA antagonist 5-(dimethylamino)-N-(3,4-dimethyl-5-isoxazolyl)-1-naphthalenesulfonamide, J. Med. Chem., 37, 329, 10.1021/jm00029a001
Suzuki, 1990, A sandwich-type enzyme immunoassay to detect immunoreactive big-endothelin-1 in plasma, J. Immunol. Meth., 127, 165, 10.1016/0022-1759(90)90065-4
Takahashi, 1993, Purification and characterization of endothelin-converting enzyme from rat lung, J. Biol. Chem., 268, 21395, 10.1016/S0021-9258(19)36936-4
Tsurumi, 1994, WS79089A, B and C, new endothelin converting enzyme inhibitors isolated from Streptosporangium roseum NO. 79089, J. Antibiotics, 47, 667, 10.7164/antibiotics.47.619
Turner, 1993, Endothelin-converting enzymes and other families of metallo-endopeptidases, Biochem. Soc. Trans., 21, 697, 10.1042/bst0210697
Ujiie, 1992, Messenger RNA expression and synthesis of endothelin-1 along rat nephron segments, J. Clin. Invest., 90, 1043, 10.1172/JCI115918
Vane, 1992, Secretory functions of the vascular endothelium, J. Physiol. Pharmacol., 43, 195
Vijayaraghavan, 1990, The hydrolysis of endothelins by neutral endopeptidase 24.11 (enkephalinase), J. Biol. Chem., 265, 14150, 10.1016/S0021-9258(18)77280-3
Waxman, 1993, Identification and characterization of endothelin converting activity from EAHY 926 cells: evidence for the physiologically relevant human enzymes, Arch. Biochem. Biophys., 308, 240, 10.1006/abbi.1994.1034
Yanagisawa, 1994, The endothelin system: a new target for therapeutic intervention, Circulation, 89, 1320, 10.1161/01.CIR.89.3.1320