EZH2 inhibition as a therapeutic strategy for lymphoma with EZH2-activating mutations

Nature - Tập 492 Số 7427 - Trang 108-112 - 2012
Michael T. McCabe1, Heidi M. Ott1, Gopinath Ganji1, Susan Korenchuk1, Christine Thompson1, Glenn S. Van Aller1, Yan Liu1, Alan P. Graves2, Anthony Della Pietra1, Elsie Diaz2, Louis V. LaFrance1, Mark Mellinger1, Céline Duquenne1, Xinrong Tian1, Ryan G. Kruger1, Charles F. McHugh1, Martín Brandt2, William H. Miller1, Dashyant Dhanak1, Sharad K. Verma1, Peter J. Tummino1, Caretha L. Creasy1
1Cancer Epigenetics Discovery Performance Unit, Cancer Research, Oncology R&D, GlaxoSmithKline, 1250 S. Collegeville Road, Collegeville, USA
2Platform Technology and Sciences, GlaxoSmithKline, 1250 S. Collegeville Road, Collegeville, USA

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