Structure−Activity Relationships for a Series of Quinoline-Based Compounds Active against Replicating and Nonreplicating <i>Mycobacterium tuberculosis</i>

Journal of Medicinal Chemistry - Tập 52 Số 7 - Trang 2109-2118 - 2009
Annamaria Lilienkampf1, Jialin Mao1, Baojie Wan1, Yuehong Wang1, Scott G. Franzblau1, Alan P. Kozikowski1
1Drug Discovery Program, Department of Medicinal Chemistry and Pharmacognosy, College of Pharmacy, University of Illinois at Chicago, 833 South Wood Street, Chicago, Illinois 60612, Institute for Tuberculosis Research, College of Pharmacy, University of Illinois at Chicago, 833 South Wood Street, Chicago, Illinois 60612

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World Health Organization, 2008, Global Tuberculosis Control: Surveillance, Planning, and Financing; WHO Report 008

Spigelman M. K., 2007, J. Infect. Dis., 196, S28−S34, 10.1086/518663

Janin Y. L., 2007, Bioorg. Med. Chem., 15, 2479, 10.1016/j.bmc.2007.01.030

Boshoff H. I. M., 2005, Nat. Rev. Microbiol., 3, 70, 10.1038/nrmicro1065

Wayne L. G., 2001, Annu. Rev. Microbiol., 55, 139, 10.1146/annurev.micro.55.1.139

Rae J. M., 2001, J. Pharmacol. Exp. Ther., 299, 849

Nayyar A., 2006, Bioorg. Med. Chem., 14, 847, 10.1016/j.bmc.2005.09.018

Jain R., 2003, Bioorg. Med. Chem. Lett., 13, 1051, 10.1016/S0960-894X(03)00074-X

Monga V., 2004, Bioorg. Med. Chem., 12, 6465, 10.1016/j.bmc.2004.09.017

Moadebi S., 2007, Drugs, 67, 2077, 10.2165/00003495-200767140-00007

Drlica K., 1999, Curr. Opin. Microbiol., 2, 504, 10.1016/S1369-5274(99)00008-9

Wang J.-Y., 2007, J. Antimicrob. Chemother., 59, 860, 10.1093/jac/dkm061

Escribano I., 2007, Chemotherapy, 53, 397, 10.1159/000109769

Andries K., 2005, Science, 307, 223, 10.1126/science.1106753

Jayaprakash S., 2006, ChemMedChem, 1, 593, 10.1002/cmdc.200600010

Mao J., 2007, ChemMedChem, 2, 1624, 10.1002/cmdc.200700112

Mao J., 2007, ChemMedChem, 2, 811, 10.1002/cmdc.200700048

Liu, W.; Dragan, V.; Strong, H. L.; Wu, Y.; Wen, Z.; Liang, J. K.; Durutlic, H.; Sutherland, Karen, W.; Pilcher, A. S.Process for preparation of 8-piperazinyl-quinoline derivativesPCT Int. Appl. WO2007146072A2, 2007.

Micetich R. G., 1985, Heterocycles, 23, 571, 10.3987/R-1985-03-0571

Lee C. B., 2001, J. Am. Chem. Soc., 123, 5249, 10.1021/ja010039j

Charbonniere L., 2006, Chem.—Eur. J., 13, 346, 10.1002/chem.200600915

Dan A., 2005, Bioorg. Med. Chem. Lett., 15, 4085, 10.1016/j.bmcl.2005.06.016

Franzblau S. G., 1998, J. Clin. Microbiol., 36, 362, 10.1128/JCM.36.2.362-366.1998

Cho S. H., 2007, Antimicrob. Agents Chemother., 51, 1380, 10.1128/AAC.00055-06

Tangallapally R. P., 2007, Curr. Top. Med. Chem., 7, 509, 10.2174/156802607780059772

Tangallapally R. P., 2005, J. Med. Chem., 48, 8261, 10.1021/jm050765n

De Angelis I., 1999, Xenobiotica, 29, 1157, 10.1080/004982599238029

Moreno S. N. J., 1985, Environ. Health Perspect., 64, 199, 10.1289/ehp.8564199

Koul A., 2007, Nat. Chem. Biol., 3, 323, 10.1038/nchembio884

Martin-Galiano A. J., 2002, Antimicrob. Agents Chemother., 46, 1680, 10.1128/AAC.46.6.1680-1687.2002

Soellner M. B., 2007, J. Am. Chem. Soc., 129, 9613, 10.1021/ja0727520

Singh R., 2003, Mol. Microbiol., 50, 751, 10.1046/j.1365-2958.2003.03712.x