The 4-N-acyl and 4-N-alkyl gemcitabine analogues with silicon-fluoride-acceptor: Application to 18F-Radiolabeling

European Journal of Medicinal Chemistry - Tập 148 - Trang 314-324 - 2018
Cesar Gonzalez1, Andersson Sanchez1, Jeffrey Collins2, Ksenia Lisova2,3, Jason T. Lee2, R. Michael van Dam2,3, M. Alejandro Barbieri4, Cheppail Ramachandran5, Stanislaw F. Wnuk6
1Department of Chemistry and Biochemistry, Florida International University, Miami, FL 33199, United States
2Crump Institute for Molecular Imaging, Department of Molecular and Medical Pharmacology, David Geffen School of Medicine, UCLA, Los Angeles, CA, 90095, United States
3Physics & Biology in Medicine Interdepartmental Graduate Program, David Geffen School of Medicine, UCLA, Los Angeles, CA, 90095, United States
4Department of Biological Sciences, Florida International University, Miami, FL, 33199, United States
5Nicklaus Children's Hospital, Miami, FL, 33155, United States
6Department of Chemistry and Biochemistry, Florida International University, Miami, FL, 33199, United States

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