Enhancement of dissolution rate of poorly-soluble active ingredients by supercritical fluid processes

Charoenchaitrakool, M., Dehghani, F., Foster, N.R., Chan, H.K., 2000. Micronization by RESS to enhance the dissolution rates of poorly water soluble pharmaceuticals. In: Eckert, C., Teja, A. (Eds.), Proceedings (CD-ROM) of the Fifth International Symposium on Supercritical Fluids.

Crison, 2000, Biopharmaceutical aspects of water-insoluble drugs for oral delivery, 97

Cristini, F., Delalonde, M., Joussot-Dubien, C., Bataille, B., 2003. Elaboration of ibuprofen microcomposites in supercritical CO2. In: Brunner, G., Kikic, I., Perrut, M. (Eds.), Proceedings of the Sixth International Symposium on Supercritical Fluid, pp. 1917–1922.

Foster, N.R., Bezanehtak, K., Charoenchaitrakool, M., Combes, G., Dehghani, F., Sze Tu, L., Thiering, R., Warwick, B., Butsami, R., Chan, H.K., (2000), Processing pharmaceuticals using dense gas technology. In: Eckert, C., Teja, A. (Eds.), Proceedings (CD-ROM) of the Fifth International Symposium on Supercritical Fluids.

Foster, 2003, Application of dense gas techniques for the production of fine particles, AAPS Pharm. Sci., 5, 105, 10.1208/ps050211

Frank, S.G., Ye, C., 2000. Small particle formation and dissolution rate enhancement of relatively insoluble drugs using rapid expansion of supercritical solutions (RESS) processing. In: Eckert, C., Teja, A. (Eds.), Proceedings (CD-ROM) of the Fifth International Symposium on Supercritical Fluids.

Gerard, 1986, 226

Higuchi, 1985

Jiang, S.Y., Chen, M., Zhao, Y.P., 2003. A study on micronization of phytosterol by the RESS technique with supercritical CO2. In: Brunner, G., Kikic, I., Perrut, M. (Eds.), Proceedings of the Sixth International Symposium on Supercritical Fluid, pp. 653–1658.

Jung, 2001, Particle design using supercritical fluids: literature and patent survey, J. Supercrit. Fluids, 20, 179, 10.1016/S0896-8446(01)00064-X

Kikic, 2000, Improvement of carbamazepine dissolution characteristics using supercritical carbon dioxide, 95

Kikic, 2002, Supercritical anti-solvent precipitation processes: different ways for improving the performances of drugs, vol. 2, 821

Knez, 2000, Micronization of pharmaceuticals using supercritical fluids, 1

Liu, 2000

Loth, 1986, Properties and dissolution of drugs micronized by crystallization from supercritical gases, Int. J. Pharm., 32, 265, 10.1016/0378-5173(86)90188-2

Martin, 2000, Nanoscale particles for pharmaceutical purpose by rapid expansion of supercritical solutions (RESS). Part II: Characterization of the product and use, 53

Perrut, M., Jung, J., Leboeuf, F., (2002). Solid state morphology of particles prepared by a supercritical fluid process. In: Venice, Bertucco, A. (Eds.), Proceedings of the Fourth International Symposium on High Pressure Process Technology and Chemical Engineering, pp. 711–716.

Perrut, 2003, Supercritical fluids applications in the pharmaceutical industry, STP Pharm. Sci., 13, 83

Perrut, 2003, Supercritical fluid formulation: process choice and scale-up, Ind. Eng. Chem. Res., 42, 6375, 10.1021/ie030144x

Perrut, 2005, Enhancement of dissolution rate of poorly-soluble active ingredients by supercritical fluid processes. Part II: Preparation of composite particles, Int. J. Pharm., 288, 11, 10.1016/j.ijpharm.2004.09.008

Prentis, 1999, Pharmaceutical innovations in the seven UK-owned pharmaceutical companies (1964–1985), Br. J. Clin. Pharmacol., 25, 387, 10.1111/j.1365-2125.1988.tb03318.x

Turk, 2002, Micronization of pharmaceutical substances by rapid expansion of supercritical solutions (RESS): a promising method to improve bio-availability of poorly soluble pharmaceutical agents, J. Supercrit. Fluids, 22, 75, 10.1016/S0896-8446(01)00109-7

Warwick, 2002, Micronization of copper–indomethacin using gas anti-solvent processes, Ind. Eng. Chem. Res., 41, 1993, 10.1021/ie010760y

Weidner, 1994, PGSS—a new process for powder generation, 229