A Convenient Microwave-Enhanced Solid-Phase Synthesis of Difficult Peptide Sequences: Case Study of Gramicidin A and CSF114(Glc)

Springer Science and Business Media LLC - Tập 13 - Trang 203-208 - 2007
Fabio Rizzolo1,2, Giuseppina Sabatino1,2, Mario Chelli1,2, Paolo Rovero1,3, Anna Maria Papini1,2
1Laboratory of Peptide & Protein Chemistry & Biology, Polo Scientifico e Tecnologico, Università di Firenze, Sesto Fiorentino, Italy
2Dipartimento di Chimica Organica “Ugo Schiff” and CNR-ICCOM, Polo Scientifico, Università di Firenze, Sesto Fiorentino, Italy
3Dipartimento di Scienze Farmaceutiche, Università di Firenze, Sesto Fiorentino, Italy

Tóm tắt

Taking into account that microwave technology applied to SPPS is proposed as a valid support to the enhancement of efficiency of coupling reactions in short times, we compared the efficacy of a new automatic monomode microwave instrument versus a traditional automatic peptide synthesizer in the synthesis of different difficult peptide sequences. We verified that microwave-assisted solid phase synthesis is convenient, in terms of yield, purity, and time consumed to prepare two peptides which were previously shown to be difficult to obtain by conventional strategy, i.e., the antibiotic Gramicidin A and a glycopeptide.

Tài liệu tham khảo

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