The Influence of Spray-Drying Parameters on Phase Behavior, Drug Distribution, and In Vitro Release of Injectable Microspheres for Sustained Release
Tài liệu tham khảo
Twaites, 2005, Synthetic polymers as drugs and therapeutics, J Mater Chem, 15, 441, 10.1039/B410799N
Rhee, 2011, Sustained-release delivery of octreotide from biodegradable polymeric microspheres, AAPS Pharm SciTech, 12, 1293, 10.1208/s12249-011-9693-z
Eerdekens, 2004, Pharmacokinetics and tolerability of long-acting risperidone in schizophrenia, Schizophr Res, 70, 91, 10.1016/j.schres.2003.11.001
Meeus, 2012, Nanoscale surface characterization and miscibility study of a spray-dried injectable polymeric matrix consisting of poly(lactic-co-glycolic acid) and polyvinylpyrrolidone, J Pharm Sci, 101, 3473, 10.1002/jps.23131
Meeus, 2013, Surface characteristics of a spray-dried polymeric matrix consisting of PLGA and PVP: Relating the influence of temperature and humidity to the thermal characteristics of these polymers, Mol Pharm, 10, 3213, 10.1021/mp400263d
Vehring, 2008, Pharmaceutical particle engineering via spray drying, Pharm Res, 25, 999, 10.1007/s11095-007-9475-1
Cal, 2010, Spray drying technique. I: Hardware and process parameters, J Pharm Sci, 99, 575, 10.1002/jps.21886
Paudel, 2013, Manufacturing of solid dispersions of poorly water soluble drugs by spray drying: Formulation and process considerations, Int J Pharm, 453, 253, 10.1016/j.ijpharm.2012.07.015
Nandiyanto, 2011, Progress in developing spray- drying methods for the production of controlled morphology particles: From the nanometer to submicrometer size ranges, Adv Powder Tech- nol, 22, 1, 10.1016/j.apt.2010.09.011
Elversson, 2003, Droplet and particle size relationship and shell thickness of inhal- able lactose particles during spray drying, J Pharm Sci, 92, 900, 10.1002/jps.10352
Wan, 2013, Critical solvent properties affecting the particle formation process and characteristics of celecoxib-loaded PLGA microparticles via spray-drying, Pharm Res, 30, 1065, 10.1007/s11095-012-0943-x
Paudel, 2012, Influence of solvent composition on the miscibility and physical stability of naproxen/PVP K 25 solid dispersions prepared by cosolvent spray-drying, Pharm Res, 29, 251, 10.1007/s11095-011-0539-x
Paudel, 2013, An investigation into the effect of spray drying temperature and atomizing conditions on miscibility, physical stability, and performance of naproxen-PVP K 25 solid dispersions, J Pharm Sci, 102, 1249, 10.1002/jps.23459
Rizi, 2011, Production of pH-responsive microparticles by spray drying: investigation of experimental parameter effects on morphological and release properties, J Pharm Sci, 100, 566, 10.1002/jps.22291
Friesen, 2002, Hydroxypropyl methylcellulose acetate succinate- based spray-dried dispersions: An overview, Mol Pharm, 5, 1003, 10.1021/mp8000793
Craig, 2002, The mechanisms of drug release from solid dispersions in water-soluble polymers, Int J Pharm, 231, 131, 10.1016/S0378-5173(01)00891-2
Siepmann, 2004, Effect of the size of biodegradable microparticles on drug release: Experiment and theory, J Control Release, 96, 123, 10.1016/j.jconrel.2004.01.011
Berkland, 2003, PLG microsphere size controls drug release rate through several competing factors, Pharm Res, 20, 1055, 10.1023/A:1024466407849
Klose, 2006, How porosity and size affect the drug release mechanisms from PLGA- based microparticles, Int J Pharm, 314, 198, 10.1016/j.ijpharm.2005.07.031
Pikal, 2004, Evaluation of glassy-state dynamics from the width of the glass transition: Results from theoretical simulation of differential scanning calorimetry and comparisons with experiment, J Pharm Sci, 93, 981, 10.1002/jps.10582
Bruning, 1996, Fragility of glass-forming systems and the width of the glass transition, J Non-Cryst Solids, 205–207, 480, 10.1016/S0022-3093(96)00264-5
Savin, 2004, Effect of the composition on the width of the calorimetric glass transition in polymer-solvent and solvent-solvent mixtures, J Polym Sci Part B: Polym Phys, 42, 1155, 10.1002/polb.10776
Kaerger, 2004, Influence of particle size and shape on flowability and compactibility of binary mixtures of paracetamol and microcrystalline cellulose, Eur J Pharm Sci, 22, 173, 10.1016/j.ejps.2004.03.005
Guo, 1985, A simple relationship between particle shape effects and density, flow rate and Hausner ratio, Powder Technol, 43, 279, 10.1016/0032-5910(85)80009-7
Fu, 2012, Effect of particle shape and size on flow properties of lactose powders, Particuology, 10, 203, 10.1016/j.partic.2011.11.003
Bodmeier, 1988, Solvent selection in the preparation of poly(D, L-lactide) microspheres prepared by the solvent evaporation method, Int J Pharm, 43, 179, 10.1016/0378-5173(88)90073-7
Dunn, 1990
Shard, 1997, XPS and SSIMS analysis revealing surface segregation and short-range order in solid films of block copolymers of PEO and PLGA, Macromolecules, 30, 3051, 10.1021/ma9519021
Opdahl, 2002, Surface segregation of methyl side branches monitored by sum frequency geeneration (SGF) vibrational spectroscopy for a series of random poly(ethylene- co-propylene) copolymers, J Phys Chem B, 106, 5212, 10.1021/jp013741a
Wang, 2001, Different surface restructuring behaviors of poly(methacrylate)s detected by SGF in water, J Am Chem Soc, 123, 9470, 10.1021/ja0164071
Thanki, 2006, Surface characteristics of PLA and PLGA films, Appl Surface Sci, 253, 2758, 10.1016/j.apsusc.2006.05.047
Verheyen, 2002, Mechanism of increased dissolution of diazepam and temazepam from polyethylene glycol 6000 solid dispersions, Int J Pharm, 249, 45, 10.1016/S0378-5173(02)00532-X
Andersson, 2013, Effects of molecular weight on permeability and microstructure of mixed ethyl-hydroxypropyl-cellulose films, Eur J Pharm Sci, 48, 240, 10.1016/j.ejps.2012.11.003