Structure–activity based study of the Smac-binding pocket within the BIR3 domain of XIAP

Bioorganic & Medicinal Chemistry - Tập 15 - Trang 2935-2943 - 2007
Aislyn D. Wist1, Lichuan Gu2, Stefan J. Riedl2, Yigong Shi2, George L. McLendon1
1Department of Chemistry, Princeton University, Princeton, NJ 08544, USA
2Department of Molecular Biology, Princeton University, Princeton, NJ 08544, USA

Tài liệu tham khảo

Green, 1998, Science, 281, 1309, 10.1126/science.281.5381.1309 Shi, 2001, Nat. Struct. Biol., 8, 394, 10.1038/87548 Thompson, 1995, Science., 267, 1456, 10.1126/science.7878464 Deveraux, 1999, Gene Dev., 13, 239, 10.1101/gad.13.3.239 LaCasse, 1998, Oncogene, 17, 3247, 10.1038/sj.onc.1202569 Du, 2000, Cell, 102, 33, 10.1016/S0092-8674(00)00008-8 Verhagen, 2000, Cell, 102, 43, 10.1016/S0092-8674(00)00009-X Ekert, 2001, J. Cell Biol., 152, 483, 10.1083/jcb.152.3.483 Srinivasula, 2001, Nat. Struct. Biol., 410, 112 Tamm, 2000, Clin. Cancer Res., 6, 1796 Archakov, 2003, Proteomics, 3, 380, 10.1002/pmic.200390053 Schade, 2005, Curr. Opin. Drug Discovery Dev., 8, 365 Liu, 2000, Nat. Struct. Biol., 408, 1004 Wu, 2000, Nat. Struct. Biol., 408, 1008 Oost, 2004, J. Med. Chem., 47, 4417, 10.1021/jm040037k Li, 2004, Science, 305, 1471, 10.1126/science.1098231 Sun, 2004, J. Am. Chem. Soc., 2004, 51 Zobel, 2006, ACS Chem. Biol., 1, 525, 10.1021/cb600276q Kipp, 2002, Biochemistry, 41, 7344, 10.1021/bi0121454 DeLano, W. The PyMol Molecular Graphics System. DeLano Scientific LLC: San Carlos, CA, USA, <http://www.pymol.org.>. Arnt, 2002, J. Biol. Chem., 277, 44236, 10.1074/jbc.M207578200 Fulda, 2002, Nat. Med., 8, 808, 10.1038/nm735 Yang, 2003, Cancer Res., 63, 831 Wipf, 1992, Tetrahedron Lett., 33, 907, 10.1016/S0040-4039(00)91572-7 Williams, 1997, Tetrahedron Lett., 38, 331, 10.1016/S0040-4039(96)02344-1