[D-Pen2,D-Pen5]enkephalin (DPDPE): a δ-selective enkephalin with low affinity for μ1 opiate binding sites

European Journal of Pharmacology - Tập 128 Số 3 - Trang 303-304 - 1986
Janet A. Clark1,2, Yossef Itzhak1,2, Victor J. Hruby3, Henry I. Yamamura4, Gavril W. Pasternak
1(Cornell University
2Memorial Sloan Kettering Cancer Center
3Chemistry and Biochemistry
4University of Arizona

Tóm tắt

Từ khóa


Tài liệu tham khảo

Goodman, 1985, Regional differences in mu1 binding of 3H-DADL-enkephalin: comparisons of thalamus and cortex, Neurosci. Lett., 59, 155, 10.1016/0304-3940(85)90192-2

Mosberg, 1983, Conformationally constrained cyclic enkephalins show pronounced delta receptor selectivity, Life Sci., 32, 2565, 10.1016/0024-3205(83)90239-4

Mosberg, 1983, Bis-penicillamine enkephalins show pronounced delta opioid receptor selectivity, 80, 5871

Pasternak, 1986, Multiple mu opiate receptors, Life Sci., 38, 1889, 10.1016/0024-3205(86)90217-1

Wolozin, 1981, Classification of multiple morphine and enkephalin binding sites in the central nervous system, 78, 6181