Preparation and characterization of pH-independent sustained release tablet containing solid dispersion granules of a poorly water-soluble drug

International Journal of Pharmaceutics - Tập 415 - Trang 83-88 - 2011
Huyen Thi Thanh Tran1, Jun Bom Park1, Ki-Hyuk Hong1, Han-Gon Choi2, Hyo-Kyung Han3, Jaehwi Lee4, Kyung Taek Oh4, Beom-Jin Lee1
1Bioavailability Control Laboratory, College of Pharmacy, Kangwon National University, Chuncheon 200-701, Republic of Korea
2College of Pharmacy, Hanyang University, Ansan 426-791, Republic of Korea
3College of Pharmacy, Dongguk University, Seoul 100-715, Republic of Korea
4College of Pharmacy, Chung-Ang University, Seoul 155-756, Republic of Korea

Tài liệu tham khảo

Barra, 2000, Modified drug release from inert matrix tablets prepared from formulation of identical composition but different organizations, J. Control. Release, 65, 419, 10.1016/S0168-3659(99)00220-5 Cao, 2004, Release behavior and photo-image of nifedipine tablet coated with high viscosity grade hydroxypropylmethylcellulose: effect of coating conditions, Int. J. Pharm., 274, 107, 10.1016/j.ijpharm.2004.01.020 Chauhan, 2005, Preparation and evaluation of glibenclamide-polyglycolized glycerides solid dispersions with silicon dioxide by spray drying technique, Eur. J. Pharm. Sci., 26, 219, 10.1016/j.ejps.2005.06.005 Chopra, 2007, Release modulating hydrophilic matrix systems of losartan potassium: optimization of formulation using statistical experiment design, Eur. J. Pharm. Biopharm., 66, 73, 10.1016/j.ejpb.2006.09.001 Fujii, 2005, Preparation, characterization, and tableting of a solid dispersion of indomethacin with crospovidone, Int. J. Pharm., 293, 145, 10.1016/j.ijpharm.2004.12.018 Gupta, 2001, Enhanced drug dissolution and bulk properties of solid dispersions granulated with a surface adsorbent, Pharm. Dev. Technol., 6, 563, 10.1081/PDT-120000294 Hirasawa, 2003, Physicochemical characterization and drug release studies of nilvadipine solid dispersion using water-insoluble polymer as a carrier, Drug Dev. Ind. Pharm., 29, 339, 10.1081/DDC-120018207 Horisawa, 2000, Physical properties of solid dispersion of a nonsteroidal anti-inflammatory drug (M-5011) with Eudragit E, Drug Dev. Ind. Pharm., 26, 1271, 10.1081/DDC-100102308 Karavas, 2007, Combining SEM, TEM, and micro-Raman techniques to differentiate between the amorphous molecular level dispersions and nanodispersions of a poorly water-soluble drug within a polymer matrix, Int. J. Pharm., 340, 76, 10.1016/j.ijpharm.2007.03.037 Leonardi, 2007, Development of prednisone:polyethylene glycol 6000 fast-release tablets from solid dispersions: solid-state characterization, dissolution behavior, and formulation parameters, AAPS PharmSciTech., 8, E1, 10.1208/pt0804108 Maggi, 2000, High molecular weight polyethylene oxides (PEOs) as an alternative to HPMC in controlled release dosage forms, Int. J. Pharm., 195, 229, 10.1016/S0378-5173(99)00402-0 Maggi, 2002, Dissolution behaviour of hydrophilic matrix tablets containing two different polyethylene oxides (PEOs) for the controlled release of a water-soluble drug. Dimension study, Biomaterials, 23, 1113, 10.1016/S0142-9612(01)00223-X Rao, 2003, Design of pH-independent controlled release matrix tablets for acidic drugs, Int. J. Pharm., 252, 81, 10.1016/S0378-5173(02)00622-1 Sahoo, 2009, Formulation of sustained-release dosage form of verapamil hydrochloride by solid dispersion technique using Eudragit RLPO or Kollidone® SR, AAPS PharmSciTech., 10, 27, 10.1208/s12249-008-9175-0 Seburg, 2006, Photosensitized degradation of losartan potassium in an extemporaneous suspension formulation, J. Pharm. Biomed. Anal., 42, 411, 10.1016/j.jpba.2006.04.030 Takeuchi, 2004, Solid dispersion particles of tolbutamide prepared with fine silica particles by the spray-drying method, Powder Technol., 141, 187, 10.1016/j.powtec.2004.03.007 Tanaka, 2005, Development of novel sustained-release system, disintegration-controlled matrix tablet (DCMT) with solid dispersion granules of nilvadipine, J. Control. Release, 108, 386, 10.1016/j.jconrel.2005.08.024 Tran, 2008, Modulation of microenvironmental pH and crystallinity of ionizable telmisartan using alkalizers in solid dispersions for controlled release, J. Control. Release, 129, 59, 10.1016/j.jconrel.2008.04.001 Tran, 2009, Dissolution-modulating mechanism of alkalizers and polymers in nanoemulsifying solid dispersion containing acidic drug, Eur. J. Pharm. Biopharm., 72, 83, 10.1016/j.ejpb.2008.12.009 Tran, 2010, Dissolution-modulating mechanism of pH modifiers in solid dispersion containing weakly acidic or basic drugs with poor water solubility, Expert Opin. Drug Deliv., 7, 647, 10.1517/17425241003645910 Tran, 2010, Physicochemical principles of controlled release solid dispersion containing a poorly water-soluble drug, Ther. Deliv., 1, 51, 10.4155/tde.10.3 Yi, 2008, Formulation of a extended release tablet containing dexibuprofen, Arch. Pharm. Res., 31, 1637, 10.1007/s12272-001-2162-6 Yi, 2008, Controlled poorly soluble drug release from solid self-microemulsifying formulations with high viscosity hydroxypropylmethylcellulose, Eur. J. Pharm. Sci., 34, 274, 10.1016/j.ejps.2008.04.010