Discovery of a β-d-2′-Deoxy-2′-α-fluoro-2′-β-C-methyluridine Nucleotide Prodrug (PSI-7977) for the Treatment of Hepatitis C Virus

Journal of Medicinal Chemistry - Tập 53 Số 19 - Trang 7202-7218 - 2010
Michael J. Sofia1, Donghui Bao2, Wonsuk Chang2, Jinfa Du2, Dhanapalan Nagarathnam2, Suguna Rachakonda2, P. Ganapati Reddy2, Bruce S. Ross2, Peiyuan Wang2, Hai‐Ren Zhang2, Shalini Bansal2, Christine Espiritu2, Meg Keilman2, Angela M. Lam2, Holly M. Micolochick Steuer2, Congrong Niu2, Michaël Otto2, Phillip A. Furman2
1Pharmasset, Inc., 303A College Road East, Princeton, New Jersey 08540, USA.
2Pharmasset, Inc., 303A College Road East, Princeton, New Jersey 08540

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