Design, Synthesis, and Structure−Activity Relationships of a Series of 3-[2-(1-Benzylpiperidin-4-yl)ethylamino]pyridazine Derivatives as Acetylcholinesterase Inhibitors

Journal of Medicinal Chemistry - Tập 44 Số 17 - Trang 2707-2718 - 2001
Jean‐Marie Contreras1, Isabelle Parrot1, Wolfgang Sippl1, Yveline Rival1, Camille G. Wermuth1
1Laboratoire de Pharmacochimie de la Communication Cellulaire, UMR 7081 du CNRS, Université Louis Pasteur, Faculté de Pharmacie, 74, route du Rhin, 67401 Illkirch Cedex, France, and Institut für Pharmazeutische Chemie, Heinrich-Heine-Universität, Düsseldorf, Universitätsstr. 1, D-40225 Düsseldorf, Germany

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