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tập trung melanin (MCH) là một peptide vòng được xác định ban đầu là một hormone lưu hành 17-amino acid ở cá xương, nơi nó được tiết ra từ tuyến yên để đáp ứng với stress và các kích thích môi trường. Ở cá, MCH làm sáng màu da bằng cách kích thích sự tụ tập của melanosome, các hạt chứa sắc tố trong các tế bào melanophore, các tế bào có nguồn gốc từ ngoại bì thần kinh được tìm thấy trong vảy cá. Mặc dù cấu trúc peptide giữa cá và động vật có vú được bảo tồn cao, nhưng ở động vật có vú, MCH không có tác dụng rõ rệt lên sắc tố; thay vào đó, dựa trên một loạt các thí nghiệm dược lý và di truyền, MCH đã nổi lên như một bộ điều chỉnh quan trọng của vùng huyết não trong việc duy trì cân bằng năng lượng, ảnh hưởng đến cả hành vi ăn uống và tiêu thụ năng lượng.\u003C\u002Fjats:p>","\u003Cjats:p>Melanin-concentrating hormone (MCH) is a cyclic peptide originally identified as a 17-amino-acid circulating hormone in teleost fish, where it is secreted by the pituitary in response to stress and environmental stimuli. In fish, MCH lightens skin color by stimulating aggregation of melanosomes, pigment-containing granules in melanophores, cells of neuroectodermal origin found in fish scales. 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1983, Characterization of melanin-concentrating hormone in chum salmon pituitaries., Nature, 305, 321, 10.1038\u002F305321a0",{"doi":2755},"10.1038\u002F305321a0",{"id":24,"text":2757,"url":24,"identifiers":2758},"Hogben, 1931, The pigmentary effectro system. VI. 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acyclic analogues of melanin concentrating hormone., Life Sci, 51, 679, 10.1016\u002F0024-3205(92)90241-G",{"doi":2774},"10.1016\u002F0024-3205(92)90241-G",{"id":24,"text":2776,"url":24,"identifiers":2777},"Kawauchi, 2004, Melanin-concentrating hormone signaling systems in fish., Peptides, 25, 1577, 10.1016\u002Fj.peptides.2004.03.025",{"doi":2778},"10.1016\u002Fj.peptides.2004.03.025",{"id":24,"text":2780,"url":24,"identifiers":2781},"Holmqvist, 1991, Galanin-like immunoreactivity in the brain of teleosts: distribution and relation to substance P, vasotocin, and isotocin in the Atlantic salmon (Salmo salar)., J Comp Neurol, 306, 361, 10.1002\u002Fcne.903060302",{"doi":2782},"10.1002\u002Fcne.903060302",{"id":24,"text":2784,"url":24,"identifiers":2785},"Vaughan, 1989, Characterization of melanin-concentrating hormone from rat hypothalamus., Endocrinology, 125, 1660, 10.1210\u002Fendo-125-3-1660",{"doi":2786},"10.1210\u002Fendo-125-3-1660",{"id":24,"text":2788,"url":24,"identifiers":2789},"Nahon, 1994, The melanin-concentrating hormone: from the peptide to the gene., Crit Rev Neurobiol, 8, 221",{},{"id":24,"text":2791,"url":24,"identifiers":2792},"Jezova, 1992, Rat melanin-concentrating hormone stimulates adrenocorticotropin secretion: evidence for a site of action in brain regions protected by the blood-brain barrier., Endocrinology, 130, 1024",{},{"id":24,"text":2794,"url":24,"identifiers":2795},"Kristensen, 1998, Hypothalamic CART is a new anorectic peptide regulated by leptin., Nature, 393, 72, 10.1038\u002F29993",{"doi":2796},"10.1038\u002F29993",{"id":24,"text":2798,"url":24,"identifiers":2799},"Parkes, 1993, Contrasting actions of melanin-concentrating hormone and neuropeptide-E-I on posterior pituitary function., Ann NY Acad Sci, 680, 588, 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MCHR1 gene in human obesity., Eur J Endocrinol, 152, 851, 10.1530\u002Feje.1.01917",{"doi":3128},"10.1530\u002Feje.1.01917",{"id":24,"text":3130,"url":24,"identifiers":3131},"Hawes, 2004, Identification and characterization of single-nucleotide polymorphisms in MCH-R1 and MCH-R2., Obes Res, 12, 1327, 10.1038\u002Foby.2004.167",{"doi":3132},"10.1038\u002Foby.2004.167",{"id":24,"text":3134,"url":24,"identifiers":3135},"Gibson, 2004, Melanin-concentrating hormone receptor mutations and human obesity: functional analysis., Obes Res, 12, 743, 10.1038\u002Foby.2004.89",{"doi":3136},"10.1038\u002Foby.2004.89",{"id":24,"text":3138,"url":24,"identifiers":3139},"Handlon, 2006, Melanin-concentrating hormone-1 receptor antagonists for the treatment of obesity., J Med Chem, 49, 4017, 10.1021\u002Fjm058239j",{"doi":3140},"10.1021\u002Fjm058239j",{"id":24,"text":3142,"url":24,"identifiers":3143},"Palani, 2005, Biaryl ureas as potent and orally efficacious melanin concentrating hormone receptor 1 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Physiological properties of hypothalamic MCH neurons identified with selective expression of reporter gene after recombinant virus infection., Neuron, 42, 635, 10.1016\u002FS0896-6273(04)00251-X",{"doi":3159},"10.1016\u002FS0896-6273(04)00251-X",{"id":24,"text":3161,"url":24,"identifiers":3162},"Eggermann, 2003, The wake-promoting hypocretin-orexin neurons are in an intrinsic state of membrane depolarization., J Neurosci, 23, 1557, 10.1523\u002FJNEUROSCI.23-05-01557.2003",{"doi":3163},"10.1523\u002FJNEUROSCI.23-05-01557.2003",{"id":24,"text":3165,"url":24,"identifiers":3166},"Bayer, 2005, Opposite effects of noradrenaline and acetylcholine upon hypocretin\u002Forexin versus melanin concentrating hormone neurons in rat hypothalamic slices., Neuroscience, 130, 807, 10.1016\u002Fj.neuroscience.2004.10.032",{"doi":3167},"10.1016\u002Fj.neuroscience.2004.10.032",{"id":24,"text":3169,"url":24,"identifiers":3170},"Burdakov, 2005, Physiological changes in glucose differentially modulate the 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10.1523\u002FJNEUROSCI.23-01-00007.2003",{"doi":3195},"10.1523\u002FJNEUROSCI.23-01-00007.2003",{"id":24,"text":3197,"url":24,"identifiers":3198},"Gonzalez, 1997, Stimulatory effect of melanin-concentrating hormone on luteinising hormone release., Neuroendocrinology, 66, 254, 10.1159\u002F000127246",{"doi":3199},"10.1159\u002F000127246",{"id":24,"text":3201,"url":24,"identifiers":3202},"Williamson-Hughes, 2005, Melanin concentrating hormone (MCH): a novel neural pathway for regulation of GnRH neurons., Brain Res, 1041, 117, 10.1016\u002Fj.brainres.2004.11.066",{"doi":3203},"10.1016\u002Fj.brainres.2004.11.066",{"id":24,"text":3205,"url":24,"identifiers":3206},"Murray, 2000, The effect of leptin on luteinizing hormone release is exerted in the zona incerta and mediated by melanin-concentrating hormone., J Neuroendocrinol, 12, 1133, 10.1046\u002Fj.1365-2826.2000.00577.x",{"doi":3207},"10.1046\u002Fj.1365-2826.2000.00577.x",{"id":24,"text":3209,"url":24,"identifiers":3210},"Chiocchio, 2001, Melanin-concentrating hormone stimulates the release of luteinizing hormone-releasing hormone and gonadotropins in the female rat acting at both median eminence and pituitary levels., Biol Reprod, 64, 1466, 10.1095\u002Fbiolreprod64.5.1466",{"doi":3211},"10.1095\u002Fbiolreprod64.5.1466",{"id":24,"text":3213,"url":24,"identifiers":3214},"Kennedy, 2001, Melanin-concentrating hormone (MCH) suppresses thyroid stimulating hormone (TSH) release, in vivo and in vitro, via the hypothalamus and the pituitary., Endocrinology, 142, 3265, 10.1210\u002Fendo.142.7.8374",{"doi":3215},"10.1210\u002Fendo.142.7.8374",{"id":24,"text":3217,"url":24,"identifiers":3218},"Kennedy, 2003, Effect of direct injection of melanin-concentrating hormone into the paraventricular nucleus: further evidence for a stimulatory role in the adrenal axis via SLC-1., J Neuroendocrinol, 15, 268, 10.1046\u002Fj.1365-2826.2003.00997.x",{"doi":3219},"10.1046\u002Fj.1365-2826.2003.00997.x",{"id":24,"text":3221,"url":24,"identifiers":3222},"Gonzalez, 1998, Behavioral effects of neuropeptide E-I (NEI) in the female rat: interactions with α-MSH, MCH and dopamine., Peptides, 19, 1007, 10.1016\u002FS0196-9781(98)00045-X",{"doi":3223},"10.1016\u002FS0196-9781(98)00045-X",{"id":24,"text":3225,"url":24,"identifiers":3226},"Sanchez, 1997, Melanin-concentrating hormone (MCH) antagonizes the effects of α-MSH and neuropeptide E-I on grooming and locomotor activities in the rat., Peptides, 18, 393, 10.1016\u002FS0196-9781(96)00327-0",{"doi":3227},"10.1016\u002FS0196-9781(96)00327-0",{"id":24,"text":3229,"url":24,"identifiers":3230},"Marsh, 2002, Melanin-concentrating hormone 1 receptor-deficient mice are lean, hyperactive, and hyperphagic and have altered metabolism., Proc Natl Acad Sci USA, 99, 3240, 10.1073\u002Fpnas.052706899",{"doi":3231},"10.1073\u002Fpnas.052706899",{"id":24,"text":3233,"url":24,"identifiers":3234},"Chen, 2002, Targeted disruption of the melanin-concentrating hormone receptor-1 results in hyperphagia and resistance to diet-induced obesity., Endocrinology, 143, 2469, 10.1210\u002Fendo.143.7.8903",{"doi":3235},"10.1210\u002Fendo.143.7.8903",{"id":24,"text":3237,"url":24,"identifiers":3238},"Zhou, 2005, Enhanced running wheel activity of both Mch1r- and Pmch-deficient mice., Regul Pept, 124, 53, 10.1016\u002Fj.regpep.2004.06.026",{"doi":3239},"10.1016\u002Fj.regpep.2004.06.026",{"id":24,"text":3241,"url":24,"identifiers":3242},"Kokkotou, 2005, Mice with MCH ablation resist diet-induced obesity through strain-specific mechanisms, Am J Physiol Regul Integr Comp Physiol, 289, R117, 10.1152\u002Fajpregu.00861.2004",{"doi":3243},"10.1152\u002Fajpregu.00861.2004",{"id":24,"text":3245,"url":24,"identifiers":3246},"Georgescu, 2005, The hypothalamic neuropeptide melanin-concentrating hormone acts in the nucleus accumbens to modulate feeding behavior and forced-swim performance., J Neurosci, 25, 2933, 10.1523\u002FJNEUROSCI.1714-04.2005",{"doi":3247},"10.1523\u002FJNEUROSCI.1714-04.2005",{"id":24,"text":3249,"url":24,"identifiers":3250},"Smith, 2005, Mesolimbic dopamine super-sensitivity in melanin-concentrating hormone-1 receptor-deficient mice., J Neurosci, 25, 914, 10.1523\u002FJNEUROSCI.4079-04.2005",{"doi":3251},"10.1523\u002FJNEUROSCI.4079-04.2005",{"id":24,"text":3253,"url":24,"identifiers":3254},"Monzon, 1999, Response to novelty after i.c.v. injection of melanin-concentrating hormone (MCH) in rats., Physiol Behav, 67, 813, 10.1016\u002FS0031-9384(99)00117-1",{"doi":3255},"10.1016\u002FS0031-9384(99)00117-1",{"id":24,"text":3257,"url":24,"identifiers":3258},"Kela, 2003, Behavioural analysis of melanin-concentrating hormone in rats: evidence for orexigenic and anxiolytic properties., Regul Pept, 114, 109, 10.1016\u002FS0167-0115(03)00114-9",{"doi":3259},"10.1016\u002FS0167-0115(03)00114-9",{"id":24,"text":3261,"url":24,"identifiers":3262},"Roy, 2006, Genetic inactivation of melanin-concentrating hormone receptor subtype 1 (MCHR1) in mice exerts anxiolytic-like behavioral effects., Neuropsychopharmacology, 31, 112, 10.1038\u002Fsj.npp.1300805",{"doi":3263},"10.1038\u002Fsj.npp.1300805",{"id":24,"text":3265,"url":24,"identifiers":3266},"Hervieu, 1995, Pro-melanin concentrating hormone messenger ribonucleic acid and peptides expression in peripheral tissues of the rat., Neuroendocrinology, 61, 348, 10.1159\u002F000126857",{"doi":3267},"10.1159\u002F000126857",{"id":24,"text":3269,"url":24,"identifiers":3270},"Verlaet, 2002, Human immune cells express ppMCH mRNA and functional MCHR1 receptor., FEBS Lett, 527, 205, 10.1016\u002FS0014-5793(02)03232-5",{"doi":3271},"10.1016\u002FS0014-5793(02)03232-5",{"id":24,"text":3273,"url":24,"identifiers":3274},"Hoogduijn, 2002, Melanin-concentrating 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