Discovery of 5-[5-Fluoro-2-oxo-1,2- dihydroindol-(3<i>Z</i>)-ylidenemethyl]-2,4- dimethyl-1<i>H</i>-pyrrole-3-carboxylic Acid (2-Diethylaminoethyl)amide, a Novel Tyrosine Kinase Inhibitor Targeting Vascular Endothelial and Platelet-Derived Growth Factor Receptor Tyrosine Kinase

Journal of Medicinal Chemistry - Tập 46 Số 7 - Trang 1116-1119 - 2003
Li Sun1, Chris Liang1, Sheri Shirazian1, Yong Zhou1, Todd Miller1, Jean Cui1, Juri Y. Fukuda1, Ji-Yu Chu1, Asaad Nematalla1, Xueyan Wang1, Hui Chen1, Anand Sistla1, Tony C. Luu1, Flora Tang1, James Cheng‐Chung Wei1, Cho Tang1
1SUGEN, Inc., 230 E. Grand Avenue, South San Francisco, California 94080

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